SCHEMBL28448730

SCHEMBL28448730

Cc1ccc(N)cc1OC(=O)CC(C)CNC(=O)OC(C)(C)C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 4/20 0.41
MAPT P10636 3/20 0.40
HPGD P15428 3/20 0.40
ALDH1A1 P00352 3/20 0.40
TSHR P16473 2/20 0.40
PCSK9 Q8NBP7 1/20 0.39
LMNA P02545 2/20 0.39
HSD17B10 Q99714 2/20 0.39
KDM4E B2RXH2 1/20 0.39
GLA P06280 1/20 0.39
GAA P10253 1/20 0.39
CASP1 P29466 1/20 0.39
RAB9A P51151 1/20 0.39
CASP7 P55210 1/20 0.39
ADRB2 P07550 1/20 0.38
ADRB1 P08588 1/20 0.38
ADRB3 P13945 1/20 0.38
ALOX15 P16050 1/20 0.37
MAPK1 P28482 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28442495 0.89 AAK1 (0.39) AAK1MAPTHPGDALDH1A1TSHR
SCHEMBL61961 0.85 ALDH1A1 (0.52) AAK1MAPTHPGDALDH1A1TSHR
SCHEMBL28520580 0.85 CYP2D6 (0.40) AAK1MAPTHPGDALDH1A1TSHR
SCHEMBL28216105 0.83 AAK1 (0.42) AAK1MAPTHPGDALDH1A1TSHR
SCHEMBL16971068 0.75 AAK1 (0.39) AAK1MAPTHPGDALDH1A1TSHR
SCHEMBL3423364 0.74 CYP2D6 (0.43) AAK1PCSK9GAAMEN1CYP2D6
SCHEMBL16971250 0.73 AAK1 (0.39) AAK1MAPTHPGDALDH1A1TSHR
SCHEMBL28521318 0.72 KDM4E (0.40) AAK1ALDH1A1KDM4EGAACYP2D6
SCHEMBL654820 0.71 KDM4A (0.45) HPGDALDH1A1KDM4ERAB9ABRD4
SCHEMBL18427975 0.70 AAK1 (0.50) AAK1CYP2C9SYK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111479813-A Triazolobenzazepines as vasopressin V1A receptor antagonists 吉瑞工厂 2020-07-31 CN disclosed