SCHEMBL28449192

SCHEMBL28449192

CCOC(=O)CCc1nc2cc(Br)ccc2[nH]c1=O

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 10/20 0.71
HSD17B10 Q99714 6/20 0.71
ALDH1A1 P00352 4/20 0.71
LMNA P02545 1/20 0.71
EGFR P00533 2/20 0.65
HPGD P15428 3/20 0.56
CYP1A2 P05177 1/20 0.56
CYP2C19 P33261 1/20 0.56
SMN1; SMN2 Q16637 1/20 0.54
MAPT P10636 4/20 0.53
MEN1 O00255 2/20 0.53
KMT2A Q03164 2/20 0.53
HTT P42858 1/20 0.52
MAPK1 P28482 1/20 0.47
PDE3B Q13370 1/20 0.45
PDE3A Q14432 1/20 0.45
P2RY12 Q9H244 1/20 0.45
JAK2 O60674 1/20 0.44
PAK4 O96013 1/20 0.44
NTRK1 P04629 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9615 0.88 EGFR (0.82) KDM4EHSD17B10ALDH1A1LMNAEGFR
SCHEMBL11363687 0.86 KDM4E (0.67) KDM4EHSD17B10ALDH1A1LMNAEGFR
SCHEMBL3533289 0.83 KDM4E (1.00) KDM4EHSD17B10ALDH1A1LMNAHPGD
SCHEMBL6602730 0.78 ALDH1A1 (0.49) KDM4EHSD17B10ALDH1A1LMNAEGFR
SCHEMBL12940747 0.77 HSD17B10 (0.67) KDM4EHSD17B10ALDH1A1LMNASMN1; SMN2
SCHEMBL10211609 0.76 KDM4E (0.57) KDM4EHSD17B10ALDH1A1LMNAEGFR
SCHEMBL28447306 0.76 EGFR (0.46) KDM4EHSD17B10ALDH1A1LMNAEGFR
SCHEMBL28445478 0.76 EGFR (0.46) KDM4EHSD17B10ALDH1A1LMNAEGFR
SCHEMBL15383503 0.75 KDM4E (0.84) KDM4EHSD17B10ALDH1A1LMNAHPGD
SCHEMBL12894110 0.74 KDM4E (0.54) KDM4EHSD17B10ALDH1A1LMNAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108997230-B Quinoxaline derivative with matrix metalloproteinase inhibitory activity, preparation method and application thereof 山东大学 2020-08-04 CN disclosed