SCHEMBL6602730

SCHEMBL6602730

CCOC(=O)c1nc2cc(Br)ccc2[nH]c1=O

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.49
SMN1; SMN2 Q16637 2/20 0.49
GABRA1 P14867 2/20 0.48
GABRA3 P34903 2/20 0.48
GABRB1 P18505 1/20 0.48
GABRB2 P47870 1/20 0.48
SIRT2 Q8IXJ6 1/20 0.47
TARBP2 Q15633 1/20 0.44
PDE3B Q13370 1/20 0.44
PDE3A Q14432 1/20 0.44
ADORA3 P0DMS8 3/20 0.43
EGFR P00533 1/20 0.43
HPGD P15428 2/20 0.43
JAK2 O60674 1/20 0.43
PAK4 O96013 1/20 0.43
NTRK1 P04629 1/20 0.43
LCK P06239 1/20 0.43
FYN P06241 1/20 0.43
CSF1R P07333 1/20 0.43
RET P07949 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6375213 0.87 ALDH1A1 (0.53) ALDH1A1SMN1; SMN2GABRA1GABRA3GABRB1
SCHEMBL9704059 0.85 ADORA3 (0.55) ALDH1A1SIRT2TARBP2ADORA3HPGD
SCHEMBL6604320 0.85 TSHR (0.48) ALDH1A1SMN1; SMN2GABRA1GABRA3GABRB1
SCHEMBL30623229 0.85 ADORA3 (0.55) ALDH1A1SIRT2TARBP2ADORA3HPGD
SCHEMBL9705717 0.84 SIRT2 (0.44) ALDH1A1SMN1; SMN2GABRA1GABRA3GABRB1
SCHEMBL16792659 0.83 SIRT2 (0.50) ALDH1A1SMN1; SMN2GABRA1GABRA3GABRB1
SCHEMBL9705656 0.81 KDM4E (0.50) ALDH1A1GABRA1GABRA3GABRB1GABRB2
SCHEMBL6705309 0.81 ALDH1A1 (0.46) ALDH1A1SMN1; SMN2GABRA1GABRA3GABRB1
SCHEMBL880365 0.81 ALDH1A1 (0.62) ALDH1A1SMN1; SMN2ADORA3HPGDGAA
SCHEMBL11371536 0.81 MAPT (0.48) ALDH1A1SMN1; SMN2METGRK5CDK8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1020453-B1 6,7-ASYMMETRICALLY DISUBSTITUTED QUINOXALINECARBOXYLIC ACID DERIVATIVES, ADDITION SALTS THEREOF, AND PROCESSES FOR THE PREPARATION OF BOTH KYORIN SEIYAKU KK (JP) 2004-05-19 EP disclosed
US-6348461-B1 CENTRAL NERVOUS SYSTEM ANTAGONIST WITH HETEROCYCLIC SUBSTITUENTS KYORIN PHARMACEUTICAL CO., LTD. (JP) 2002-02-19 US disclosed
EP-1020453-A1 6,7-ASYMMETRICALLY DISUBSTITUTED QUINOXALINECARBOXYLIC ACID DERI VATIVES, ADDITION SALTS THEREOF, AND PROCESSES FOR THE PREPARATION OF BOTH KYORIN PHARMACEUTICAL CO., LTD. (JP) 2000-07-19 EP disclosed