SCHEMBL28449256

SCHEMBL28449256

CC(=O)c1cn(C(C)=O)c(=O)nc1N

nearest known ligand 0.34

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.34
BRD4 O60885 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
PTPN11 Q06124 1/20 0.31
CREBBP Q92793 1/20 0.31
EEF2K O00418 1/20 0.31
NOTUM Q6P988 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5694237 0.80 EP300 (0.34) NOTUM
SCHEMBL4727065 0.79 NOTUM (0.30) NOTUM
SCHEMBL21186 0.67 NOTUM (0.43) NOTUM
SCHEMBL5694084 0.67 DNMT1 (0.37) NOTUM
SCHEMBL8228221 0.66 ADORA2A (0.38) SMN1; SMN2BRD4L3MBTL1
Methane SCHEMBL27916787 0.66 NOTUM (0.42) NOTUM
SCHEMBL19310470 0.66 GABRP (0.38) BRD4L3MBTL1
SCHEMBL27696561 0.66 EP300 (0.36)
SCHEMBL27740855 0.64 NOTUM (0.41) NOTUM
SCHEMBL19820712 0.63 GABRP (0.52) SMN1; SMN2L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111675660-B Preparation method for synthesizing palbociclib intermediate and method for synthesizing palbociclib 奥锐特药业股份有限公司 2021-12-10 CN disclosed
CN-111675660-A Preparation method for synthesizing palbociclib intermediate and method for synthesizing palbociclib 奥锐特药业股份有限公司 2020-09-18 CN disclosed