SCHEMBL28451702

SCHEMBL28451702

Clc1ccc(N2CCc3ccccc3C2CCc2ccccc2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.47
ESR2 Q92731 1/20 0.47
NR1I2 O75469 1/20 0.46
MAOA P21397 1/20 0.46
PTGS2 P35354 1/20 0.46
OPRK1 P41145 1/20 0.46
SLC6A3 Q01959 1/20 0.46
SIGMAR1 Q99720 5/20 0.42
GRIN1 Q05586 3/20 0.42
GRIN2B Q13224 3/20 0.42
TP53 P04637 1/20 0.42
TSHR P16473 1/20 0.42
MAPK1 P28482 1/20 0.42
DRD4 P21917 3/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24916731 0.90 ESR1 (0.52) ESR1ESR2SIGMAR1GRIN1GRIN2B
SCHEMBL25163185 0.90 ESR1 (0.52) ESR1ESR2SIGMAR1GRIN1GRIN2B
SCHEMBL28451558 0.87 SLC6A4 (0.47) ESR1ESR2SIGMAR1GRIN1GRIN2B
SCHEMBL28451705 0.87 OPRM1 (0.46) ESR1ESR2OPRK1SIGMAR1GRIN1
SCHEMBL28452022 0.85 ESR1 (0.45) ESR1ESR2NR1I2MAOAPTGS2
SCHEMBL28452101 0.84 MTNR1B (0.48) ESR1ESR2SIGMAR1GRIN1GRIN2B
SCHEMBL28451201 0.82 GRIN2B (0.50) ESR1ESR2SIGMAR1GRIN1GRIN2B
SCHEMBL28897568 0.82 DRD4 (0.47) ESR1ESR2OPRK1DRD4
SCHEMBL28454061 0.82 ESR1 (0.44) ESR1ESR2SIGMAR1GRIN1GRIN2B
SCHEMBL28448183 0.81 ESR1 (0.62) ESR1ESR2SIGMAR1GRIN1GRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111592563-A Compound containing carbon-silicon bond and application thereof 中国科学院上海有机化学研究所 2020-08-28 CN disclosed