SCHEMBL28454064

SCHEMBL28454064

NC(=O)Oc1ccc(-n2cc(C=O)cn2)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.43
RAB9A P51151 3/20 0.43
SMN1; SMN2 Q16637 3/20 0.43
MAPKAPK2 P49137 1/20 0.43
HDAC1 Q13547 1/20 0.38
HDAC2 Q92769 1/20 0.38
MAP4K4 O95819 1/20 0.37
KMT2A Q03164 6/20 0.36
KDM4E B2RXH2 4/20 0.36
ALDH1A1 P00352 4/20 0.36
MEN1 O00255 3/20 0.36
MAPT P10636 2/20 0.36
KCNJ1 P48048 1/20 0.36
MAPK1 P28482 1/20 0.36
HPGDS O60760 1/20 0.36
ALKBH2 Q6NS38 1/20 0.36
PARP10 Q53GL7 1/20 0.36
PARP3 Q9Y6F1 1/20 0.36
KIF11 P52732 1/20 0.35
GRM2 Q14416 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11478630 0.79 ALDH1A1 (0.52) NPC1RAB9ASMN1; SMN2MAPKAPK2KMT2A
SCHEMBL28362215 0.78 KMT2A (0.36) NPC1RAB9ASMN1; SMN2KMT2AKDM4E
SCHEMBL28450895 0.77 MAPKAPK2 (0.43) NPC1RAB9ASMN1; SMN2MAPKAPK2MAP4K4
SCHEMBL21281739 0.77 SMN1; SMN2 (0.47) NPC1RAB9ASMN1; SMN2HDAC1HDAC2
SCHEMBL15104662 0.75 RXRA (0.41) NPC1RAB9ASMN1; SMN2KDM4EALDH1A1
SCHEMBL21281737 0.75 SMN1; SMN2 (0.39) NPC1RAB9ASMN1; SMN2MAPKAPK2KDM4E
SCHEMBL10081937 0.74 KMT2A (0.58) SMN1; SMN2KMT2AKDM4EALDH1A1MEN1
SCHEMBL28358602 0.74 NPC1 (0.31) NPC1RAB9A
SCHEMBL1990298 0.73 MTOR (0.52) NPC1RAB9ASMN1; SMN2KMT2AKDM4E
SCHEMBL18586366 0.73 PTGS2 (0.47) NPC1RAB9ASMN1; SMN2HDAC1HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111601810-A Inhibitors of indoleamine 2, 3-dioxygenase and/or tryptophan 2, 3-dioxygenase 爱杜西亚药品有限公司 2020-08-28 CN disclosed