SCHEMBL28454450

SCHEMBL28454450

O=C(Nc1nnc(C2CCCO2)o1)c1ccc([N+](=O)[O-])o1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 3/20 0.49
KMT2A Q03164 6/20 0.47
MEN1 O00255 4/20 0.47
GAA P10253 3/20 0.47
GLA P06280 2/20 0.47
KDM4E B2RXH2 1/20 0.47
USP2 O75604 1/20 0.47
RXFP1 Q9HBX9 1/20 0.47
DDIT3 P35638 2/20 0.47
L3MBTL1 Q9Y468 1/20 0.45
LMNA P02545 5/20 0.45
HPGD P15428 2/20 0.45
HTT P42858 2/20 0.45
NPC1 O15118 3/20 0.44
RAB9A P51151 3/20 0.44
POLB P06746 3/20 0.44
MITF O75030 1/20 0.44
NFKB1 P19838 1/20 0.44
NFKB2 Q00653 1/20 0.44
RELA Q04206 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28452446 0.88 TDP1 (0.40) TDP1KMT2AMEN1GAAGLA
SCHEMBL28455352 0.80 NPC1 (0.60) KMT2AMEN1GAAGLAKDM4E
SCHEMBL28449547 0.79 ADCY1 (0.41) TDP1KMT2AMEN1KDM4ELMNA
SCHEMBL22594348 0.69 ADCY1 (0.53) TDP1KDM4ELMNAHTTNPC1
SCHEMBL24290767 0.68 KMT2A (0.78) KMT2AMEN1GAAGLAKDM4E
SCHEMBL7485465 0.67 DDIT3 (0.53) TDP1KMT2AMEN1GAAGLA
SCHEMBL18952982 0.67 TDP1 (0.69) TDP1KMT2AMEN1GAAGLA
SCHEMBL6432446 0.67 MITF (0.68) TDP1KMT2AMEN1DDIT3L3MBTL1
SCHEMBL1899946 0.66 STAT3 (0.64) TDP1KMT2AMEN1GAAGLA
SCHEMBL7485300 0.66 DDIT3 (0.52) KMT2AMEN1GAAGLAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109535146-B Antituberculous compound and its preparation method and use 中国医学科学院医药生物技术研究所 2020-09-22 CN disclosed