SCHEMBL28454652

SCHEMBL28454652

CCNc1c(C(N)=O)ccc(CC)c1CC

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MKNK1 Q9BUB5 1/20 0.38
MKNK2 Q9HBH9 1/20 0.38
SMN1; SMN2 Q16637 2/20 0.35
MAPT P10636 2/20 0.35
PKM P14618 1/20 0.35
MAPK1 P28482 1/20 0.35
ALDH1A1 P00352 3/20 0.35
HSD17B10 Q99714 2/20 0.35
KDM4E B2RXH2 2/20 0.35
HPGD P15428 2/20 0.35
CACNA1C Q13936 2/20 0.35
SCN5A Q14524 2/20 0.35
HSP90AA1 P07900 1/20 0.35
PARP1 P09874 1/20 0.33
SIRT2 Q8IXJ6 1/20 0.32
LRRK2 Q5S007 2/20 0.32
IKBKB O14920 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
CYP1A2 P05177 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27752032 0.85 KDM4E (0.37) SMN1; SMN2PKMALDH1A1HSD17B10KDM4E
SCHEMBL5618594 0.78 PARP1 (0.38) SMN1; SMN2MAPTALDH1A1HSD17B10KDM4E
Bromide SCHEMBL9317974 0.77 PARP1 (0.37) SMN1; SMN2MAPTALDH1A1HSD17B10KDM4E
Hydrochloric Acid SCHEMBL10630450 0.77 PARP1 (0.37) SMN1; SMN2MAPTALDH1A1HSD17B10KDM4E
SCHEMBL474164 0.75 NNMT (0.36) SMN1; SMN2MAPTPKMALDH1A1HSD17B10
SCHEMBL6607453 0.75 GABRP (0.36) SMN1; SMN2MAPTMAPK1ALDH1A1HSD17B10
SCHEMBL2161703 0.75 PARP1 (0.36) SMN1; SMN2MAPTPKMALDH1A1HSD17B10
SCHEMBL288795 0.75 ERN1 (0.40) SMN1; SMN2MAPTALDH1A1HSD17B10KDM4E
SCHEMBL28455285 0.75 CYP3A4 (0.40) MKNK1MKNK2SMN1; SMN2MAPTPKM
Hydrochloric Acid SCHEMBL6639008 0.74 GABRP (0.35) SMN1; SMN2MAPTMAPK1ALDH1A1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114516855-A Preparation of pyridylpyrazole amide compounds and intermediates therefor 湖南化工研究院有限公司 2022-05-20 CN claimed
CN-114516854-A Preparation method of 1-pyridyl pyrazole amide compound and intermediate thereof 湖南化工研究院有限公司 2022-05-20 CN claimed
CN-111662269-B 1-pyridyl pyrazole amide compound and preparation method and application thereof 湖南化工研究院有限公司 2021-05-07 CN claimed
CN-111662269-A 1-pyridyl pyrazole amide compound and preparation method and application thereof 湖南化工研究院有限公司 2020-09-15 CN claimed
CN-114516855-A Preparation of pyridylpyrazole amide compounds and intermediates therefor 湖南化工研究院有限公司 2022-05-20 CN disclosed
CN-114516854-A Preparation method of 1-pyridyl pyrazole amide compound and intermediate thereof 湖南化工研究院有限公司 2022-05-20 CN disclosed
CN-111662269-B 1-pyridyl pyrazole amide compound and preparation method and application thereof 湖南化工研究院有限公司 2021-05-07 CN disclosed
CN-111662269-A 1-pyridyl pyrazole amide compound and preparation method and application thereof 湖南化工研究院有限公司 2020-09-15 CN disclosed