SCHEMBL28455285

SCHEMBL28455285

CCNc1c(C(N)=O)ccc(C)c1C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.40
TSHR P16473 1/20 0.40
RECQL P46063 1/20 0.40
MKNK1 Q9BUB5 1/20 0.39
MKNK2 Q9HBH9 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.36
MAPT P10636 1/20 0.36
PKM P14618 1/20 0.36
MAPK1 P28482 1/20 0.36
CLCN2 P51788 1/20 0.36
SIRT3 Q9NTG7 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
HPGD P15428 1/20 0.36
HSD17B10 Q99714 1/20 0.36
CYP2D6 P10635 1/20 0.34
HSP90AA1 P07900 1/20 0.34
NNMT P40261 2/20 0.33
LRRK2 Q5S007 3/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29212433 0.82 CA12 (0.34) SMN1; SMN2MAPTPKMCLCN2SIRT3
SCHEMBL27701122 0.80 NNMT (0.42) TSHRMKNK1MKNK2MAPTPKM
SCHEMBL12289243 0.77 ALDH1A1 (0.49) MKNK2SMN1; SMN2PKMCLCN2SIRT3
SCHEMBL22788208 0.75 TSHR (0.47) CYP3A4TSHRRECQLMAPTKDM4E
SCHEMBL28454652 0.75 MKNK1 (0.38) CYP3A4MKNK1MKNK2SMN1; SMN2MAPT
SCHEMBL13451003 0.73 POLB (0.37) CYP3A4TSHRRECQLMKNK1MKNK2
SCHEMBL3698508 0.73 MYC (0.44) CYP3A4SMN1; SMN2MAPTPKMMAPK1
SCHEMBL354227 0.73 SIRT3 (0.45) TSHRMKNK1MKNK2MAPTMAPK1
SCHEMBL28202663 0.72 ALDH1A1 (0.42) CYP3A4TSHRMKNK1MKNK2SMN1; SMN2
Hydrochloric Acid SCHEMBL1776795 0.71 SIRT3 (0.44) TSHRMKNK1MKNK2MAPTMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114516855-A Preparation of pyridylpyrazole amide compounds and intermediates therefor 湖南化工研究院有限公司 2022-05-20 CN claimed
CN-114516854-A Preparation method of 1-pyridyl pyrazole amide compound and intermediate thereof 湖南化工研究院有限公司 2022-05-20 CN claimed
CN-111662269-B 1-pyridyl pyrazole amide compound and preparation method and application thereof 湖南化工研究院有限公司 2021-05-07 CN claimed
CN-111662269-A 1-pyridyl pyrazole amide compound and preparation method and application thereof 湖南化工研究院有限公司 2020-09-15 CN claimed
CN-114516855-A Preparation of pyridylpyrazole amide compounds and intermediates therefor 湖南化工研究院有限公司 2022-05-20 CN disclosed
CN-114516854-A Preparation method of 1-pyridyl pyrazole amide compound and intermediate thereof 湖南化工研究院有限公司 2022-05-20 CN disclosed
CN-111662269-B 1-pyridyl pyrazole amide compound and preparation method and application thereof 湖南化工研究院有限公司 2021-05-07 CN disclosed
CN-111662269-A 1-pyridyl pyrazole amide compound and preparation method and application thereof 湖南化工研究院有限公司 2020-09-15 CN disclosed