SCHEMBL28454697

SCHEMBL28454697

CC(=O)OCCN(CCCC#N)Cc1ccccc1

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.53
LMNA P02545 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2D6 P10635 1/20 0.43
POLB P06746 2/20 0.42
ALDH1A1 P00352 4/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
CYP3A4 P08684 1/20 0.42
MAOB P27338 5/20 0.41
CHRM1 P11229 1/20 0.40
HDAC3 O15379 2/20 0.40
HDAC1 Q13547 2/20 0.40
HDAC2 Q92769 2/20 0.40
HDAC8 Q9BY41 2/20 0.40
NCOR2 Q9Y618 2/20 0.40
CHRNB2 P17787 1/20 0.40
CHRNB4 P30926 1/20 0.40
CHRNA3 P32297 1/20 0.40
CHRNA4 P43681 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28451212 0.88 LMNA (0.44) TSHRLMNACYP1A2CYP2D6POLB
SCHEMBL12671106 0.86 TSHR (0.65) TSHRLMNACYP1A2CYP2D6POLB
SCHEMBL3223085 0.83 TSHR (0.69) TSHRLMNACYP1A2CYP2D6POLB
SCHEMBL7877735 0.82 ALDH1A1 (0.48) LMNAPOLBALDH1A1HDAC3HDAC1
SCHEMBL2945207 0.80 ALDH1A1 (0.45) LMNAPOLBALDH1A1SMN1; SMN2HDAC3
SCHEMBL10962715 0.79 POLB (0.47) POLBALDH1A1HDAC3HDAC1HDAC2
SCHEMBL154270 0.79 ALDH1A1 (0.48) POLBALDH1A1MAOBCHRM1HDAC3
SCHEMBL28664666 0.78 POLB (0.48) LMNAPOLBALDH1A1HDAC3HDAC1
SCHEMBL28562689 0.78 POLB (0.46) LMNACYP1A2CYP2D6POLBALDH1A1
SCHEMBL17508109 0.77 ALDH1A1 (0.47) POLBALDH1A1MAOBHDAC3HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111670034-A Pyranopyrazoles and pyrazolopyridines immunomodulators for the treatment of autoimmune diseases 洛克菲勒大学 2020-09-15 CN disclosed