SCHEMBL28456262

SCHEMBL28456262

CC(C)(C)OC(=O)N1CCCC(n2cc3ccc(-c4ccccc4F)cc3n2)C1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 1/20 0.41
PIK3R2 O00459 1/20 0.41
PIK3CA P42336 1/20 0.41
PIK3CB P42338 1/20 0.41
PIK3CG P48736 1/20 0.41
PIK3R5 Q8WYR1 1/20 0.41
PIK3R3 Q92569 1/20 0.41
USP30 Q70CQ3 2/20 0.41
BTK Q06187 5/20 0.40
HDAC6 Q9UBN7 2/20 0.40
HDAC4 P56524 1/20 0.40
HSD17B13 Q7Z5P4 1/20 0.40
TRPV3 Q8NET8 1/20 0.40
EGFR P00533 2/20 0.40
SRC P12931 2/20 0.40
KDM5A P29375 1/20 0.39
JAK2 O60674 1/20 0.39
JAK1 P23458 1/20 0.39
ALOX5AP P20292 1/20 0.39
FEN1 P39748 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28457726 0.93 PIK3CD (0.41) PIK3CDPIK3R2PIK3CAPIK3CBPIK3CG
SCHEMBL28458766 0.90 BTK (0.42) PIK3CDPIK3R2PIK3CAPIK3CBPIK3CG
SCHEMBL28898133 0.90 APLNR (0.44) PIK3CDPIK3R2PIK3CAPIK3CBPIK3CG
SCHEMBL28455465 0.89 HSD17B13 (0.44) BTKHSD17B13JAK2JAK1
SCHEMBL28898963 0.88 HDAC1 (0.46) USP30BTKHDAC6HDAC4JAK2
SCHEMBL28452393 0.87 HSD17B13 (0.49) PIK3CDPIK3R2PIK3CAPIK3CBPIK3CG
SCHEMBL28452589 0.87 USP30 (0.45) USP30BTKHDAC6HDAC4EGFR
SCHEMBL28456326 0.86 APLNR (0.42) PIK3CDPIK3CAPIK3CBPIK3CGUSP30
SCHEMBL28461486 0.84 GPR119 (0.46) USP30HDAC6HDAC4CHEK2
SCHEMBL28449733 0.84 CNR1 (0.46) USP30BTKHDAC6HDAC4CHEK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111662232-B Small molecule compound with 2H-indazole structure and synthesis and application thereof 中国科学院上海药物研究所 2022-08-02 CN disclosed
CN-111662232-A Small molecule compound with 2H-indazole structure and synthesis and application thereof 中国科学院上海药物研究所 2020-09-15 CN disclosed