SCHEMBL28449733

SCHEMBL28449733

CC(C)(C)OC(=O)N1CCCC(n2cc3ccc(-c4ccc(Cl)cc4)cc3n2)C1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 2/20 0.46
CNR2 P34972 2/20 0.46
USP30 Q70CQ3 1/20 0.43
BTK Q06187 2/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
GPR119 Q8TDV5 2/20 0.41
CHEK2 O96017 2/20 0.41
HDAC4 P56524 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
CACNB4 O00305 2/20 0.40
CACNA1A O00555 2/20 0.40
CACNA1G O43497 2/20 0.40
CACNG3 O60359 2/20 0.40
CACNA1F O60840 2/20 0.40
CACNA1H O95180 2/20 0.40
CACNB3 P54284 2/20 0.40
CACNA2D1 P54289 2/20 0.40
CACNG7 P62955 2/20 0.40
CACNA1B Q00975 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28460213 0.92 USP30 (0.45) CNR1CNR2USP30BTKCHEK2
SCHEMBL28898963 0.91 HDAC1 (0.46) USP30BTKGPR119CHEK2HDAC4
SCHEMBL28461486 0.91 GPR119 (0.46) USP30GPR119CHEK2HDAC4HDAC6
SCHEMBL28458581 0.90 SRC (0.47) USP30BTKMEN1KMT2AGPR119
SCHEMBL28455501 0.88 GPR119 (0.47) USP30BTKMEN1KMT2AGPR119
SCHEMBL28458766 0.88 BTK (0.42) CNR1CNR2USP30BTKCHEK2
SCHEMBL28452589 0.86 USP30 (0.45) USP30BTKGPR119CHEK2HDAC4
SCHEMBL29968466 0.86 GPR119 (0.48) USP30BTKGPR119CHEK2HDAC4
SCHEMBL28458448 0.86 GPR119 (0.48) USP30BTKGPR119CHEK2HDAC4
SCHEMBL28456256 0.85 FPR2 (0.48) USP30MEN1KMT2ACHEK2HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111662232-B Small molecule compound with 2H-indazole structure and synthesis and application thereof 中国科学院上海药物研究所 2022-08-02 CN disclosed
CN-111662232-A Small molecule compound with 2H-indazole structure and synthesis and application thereof 中国科学院上海药物研究所 2020-09-15 CN disclosed