SCHEMBL28456512

SCHEMBL28456512

Nc1ccc(Br)c(-c2ccc(F)cc2F)c1F

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.48
MEN1 O00255 1/20 0.35
POLB P06746 1/20 0.35
MAPT P10636 1/20 0.35
HTT P42858 1/20 0.35
KMT2A Q03164 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
IDO1 P14902 2/20 0.33
AGXT P21549 2/20 0.33
KIT P10721 1/20 0.33
PIK3R1 P27986 1/20 0.33
PIK3CA P42336 1/20 0.33
KEAP1 Q14145 1/20 0.33
ADORA2A P29274 2/20 0.32
CLK1 P49759 1/20 0.32
ADORA1 P30542 1/20 0.31
KDM1A O60341 2/20 0.31
KCNH2 Q12809 2/20 0.31
HTR5A P47898 1/20 0.31
ALOX15 P16050 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29765813 1.00 ALDH1A1 (0.48) ALDH1A1MEN1POLBMAPTHTT
SCHEMBL17535945 0.76 AMY1A (0.42) ALDH1A1MEN1POLBMAPTKMT2A
SCHEMBL4307951 0.74 ALDH1A1 (0.56) ALDH1A1MEN1HTTKMT2AIDO1
SCHEMBL28552674 0.73 ALDH1A1 (0.54) ALDH1A1MEN1HTTKMT2AL3MBTL1
SCHEMBL21464154 0.72 ALDH1A1 (0.52) ALDH1A1MEN1POLBMAPTKMT2A
SCHEMBL16637006 0.71 TTR (0.46) ALDH1A1MEN1MAPTKMT2AKEAP1
SCHEMBL6284436 0.71 ALDH1A1 (0.42) ALDH1A1MEN1KMT2AIDO1AGXT
SCHEMBL28920191 0.70 ALDH1A1 (0.37) ALDH1A1MAPTIDO1AGXTKIT
SCHEMBL29350499 0.70
SCHEMBL14413 0.70

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106488910-B Inhibitors of KRAS G12C 亚瑞克西斯制药公司 2020-07-31 CN disclosed