SCHEMBL28920191

SCHEMBL28920191

Nc1cc(Cl)c(-c2ccc(F)cc2F)c(Br)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.37
KIT P10721 1/20 0.35
HTR5A P47898 2/20 0.34
ALOX15 P16050 1/20 0.34
ADORA2A P29274 2/20 0.33
ADORA2B P29275 1/20 0.33
CYP3A4 P08684 2/20 0.32
GAA P10253 1/20 0.32
MAPT P10636 1/20 0.32
PIK3R1 P27986 1/20 0.32
PIK3CA P42336 1/20 0.32
IDO1 P14902 2/20 0.32
AGXT P21549 2/20 0.32
KDM1A O60341 2/20 0.31
KDM1B Q8NB78 2/20 0.31
MAPK14 Q16539 2/20 0.31
MAPK13 O15264 1/20 0.31
MAPK12 P53778 1/20 0.31
MAPK11 Q15759 1/20 0.31
TSHR P16473 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19433368 0.71 APP (0.43) ALDH1A1KITALOX15ADORA2AADORA2B
SCHEMBL29765813 0.70 ALDH1A1 (0.48) ALDH1A1KITHTR5AALOX15ADORA2A
SCHEMBL28456512 0.70 ALDH1A1 (0.48) ALDH1A1KITHTR5AALOX15ADORA2A
SCHEMBL16013714 0.68 CYP3A4 (0.39) ALDH1A1ALOX15ADORA2ACYP3A4GAA
SCHEMBL16395977 0.68 ALDH1A1 (0.41) ALDH1A1KITADORA2AIDO1AGXT
SCHEMBL14744345 0.68 RORC (0.45) ALDH1A1ADORA2ACYP3A4
SCHEMBL14747029 0.68 AR (0.38) ALDH1A1GAA
SCHEMBL29646646 0.67 ALDH1A1 (0.48) ALDH1A1KITADORA2AIDO1AGXT
SCHEMBL21819775 0.67 ALDH1A1 (0.48) ALDH1A1KITADORA2AIDO1AGXT
SCHEMBL14744163 0.67 CYP3A4 (0.42) ALDH1A1CYP3A4MAPK14MAPK13MAPK12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115490709-A KRASG12D inhibitor and application thereof in medicine 四川海思科制药有限公司 2022-12-20 CN disclosed