SCHEMBL28458688

SCHEMBL28458688

Cn1c(Cl)c(C(=O)O)cc(Br)c1=O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.38
ESR2 Q92731 1/20 0.38
LCK P06239 1/20 0.37
FYN P06241 1/20 0.37
AKR1C4 P17516 1/20 0.35
AKR1C3 P42330 1/20 0.35
AKR1C2 P52895 1/20 0.35
AKR1C1 Q04828 1/20 0.35
HSD17B10 Q99714 2/20 0.35
MYC P01106 5/20 0.35
TSHR P16473 1/20 0.34
DYRK1A Q13627 1/20 0.33
ALDH1A1 P00352 1/20 0.33
MAPK10 P53779 1/20 0.33
NOTUM Q6P988 1/20 0.33
KMT2A Q03164 1/20 0.33
NR4A1 P22736 3/20 0.33
GAA P10253 1/20 0.33
MCL1 Q07820 1/20 0.33
CTSB P07858 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL391750 0.81 ALDH1A1 (0.43) HSD17B10TSHRALDH1A1MAPK10KMT2A
SCHEMBL27926911 0.80 KDM4E (0.42) HSD17B10MYCTSHRDYRK1AALDH1A1
SCHEMBL15228293 0.80 NOTUM (0.40) ESR1ESR2LCKFYNAKR1C4
SCHEMBL15051254 0.75 LMNA (0.39) AKR1C4AKR1C3AKR1C2AKR1C1HSD17B10
SCHEMBL22470670 0.73 LCK (0.42) ESR1ESR2LCKFYNAKR1C4
SCHEMBL13560140 0.69 L3MBTL1 (0.40) HSD17B10ALDH1A1KMT2AGAA
SCHEMBL12130341 0.68 SMN1; SMN2 (0.39) MYCTSHRALDH1A1NOTUMKMT2A
SCHEMBL27794857 0.68 NOTUM (0.37) ESR1ESR2LCKFYNAKR1C4
SCHEMBL26655052 0.68 KMT2A (0.37) LCKFYNHSD17B10ALDH1A1KMT2A
SCHEMBL71146 0.66 LCK (0.60) LCKFYNAKR1C4AKR1C3AKR1C2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111704611-B Aryl spiro SHP2 inhibitor compound, preparation method and application 上海凌达生物医药有限公司 2022-01-14 CN disclosed
CN-111704611-A Aryl spiro SHP2 inhibitor compound, preparation method and application 上海凌达生物医药有限公司 2020-09-25 CN disclosed