SCHEMBL28464584

SCHEMBL28464584

CC(C)(C)OC(=O)NC(CC[O])c1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CTSK P43235 6/20 0.53
CTSS P25774 4/20 0.53
MAPT P10636 2/20 0.47
ATM Q13315 1/20 0.47
CTSL P07711 1/20 0.45
CTSB P07858 1/20 0.45
GABRB1 P18505 1/20 0.44
GABRB2 P47870 1/20 0.44
PPARA Q07869 2/20 0.44
PPARG P37231 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4353938 0.88 CTSK (0.53) CTSKCTSSMAPTATMCTSL
SCHEMBL4961187 0.88 CTSK (0.56) CTSKCTSSMAPTATMCTSL
SCHEMBL4583120 0.88 CTSK (0.53) CTSKCTSSMAPTATMCTSL
SCHEMBL56698 0.88 CTSK (0.53) CTSKCTSSMAPTATMCTSL
SCHEMBL56596 0.88 CTSK (0.53) CTSKCTSSMAPTATMCTSL
SCHEMBL19517266 0.88 CTSK (0.56) CTSKCTSSMAPTATMCTSL
SCHEMBL10324741 0.87 CTSK (0.52) CTSKCTSSMAPTATMCTSL
SCHEMBL27594478 0.87 CTSK (0.52) CTSKCTSSMAPTATMCTSL
SCHEMBL21219239 0.87 CTSK (0.52) CTSKCTSSMAPTATMCTSL
SCHEMBL6007487 0.87 CTSK (0.52) CTSKCTSSMAPTATMCTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107624113-B Tetrahydropyridopyrimidines and tetrahydropyridopyridines as inhibitors of HBsAg (HBV surface antigen) and HBV DNA production for the treatment of hepatitis B virus infection 豪夫迈·罗氏有限公司 2020-10-23 CN disclosed