SCHEMBL28466232

SCHEMBL28466232

C=C(NC(C)=O)c1ccc(CCCC)cc1

nearest known ligand 0.57

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PLK1 P53350 1/20 0.57
THRA P10827 7/20 0.56
THRB P10828 7/20 0.56
RARB P10826 4/20 0.53
TRPV1 Q8NER1 1/20 0.50
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49
POLB P06746 1/20 0.49
ALDH1A1 P00352 1/20 0.49
HPGD P15428 1/20 0.49
HSD17B10 Q99714 1/20 0.49
HAO1 Q9UJM8 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28460406 0.95 THRA (0.63) PLK1THRATHRBRARBMEN1
SCHEMBL28466726 0.90 PLK1 (0.54) PLK1THRATHRBTRPV1KMT2A
SCHEMBL28470841 0.83 ALDH1A1 (0.52) PLK1THRATHRBMEN1KMT2A
SCHEMBL28459349 0.82 TRPV1 (0.63) PLK1THRATHRBRARBTRPV1
SCHEMBL18977659 0.80 PLK1 (0.49) PLK1THRATHRBRARBTRPV1
SCHEMBL19449792 0.80 EPHX2 (0.41) PLK1THRATHRBKMT2APOLB
SCHEMBL28472389 0.79 TP53 (0.54) PLK1RARBKMT2A
SCHEMBL5382633 0.78 THRA (0.61) PLK1THRATHRBRARBTRPV1
SCHEMBL19449796 0.78 KMT2A (0.40) PLK1THRATHRBKMT2APOLB
SCHEMBL19435750 0.78 CA1 (0.48) PLK1THRATHRBMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111747904-A Polyfluoroalkenyl substituted oxazole compound and preparation method thereof 南京工业大学 2020-10-09 CN claimed
CN-111747904-A Polyfluoroalkenyl substituted oxazole compound and preparation method thereof 南京工业大学 2020-10-09 CN disclosed