SCHEMBL28459349

SCHEMBL28459349

C=C(NC(=O)c1ccc(CCCC)cc1)c1ccccc1

nearest known ligand 0.63

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 2/20 0.63
PLK1 P53350 5/20 0.63
HDAC8 Q9BY41 1/20 0.51
RARB P10826 1/20 0.51
PLK3 Q9H4B4 3/20 0.51
TMEM97 Q5BJF2 1/20 0.51
SIGMAR1 Q99720 1/20 0.51
HDAC1 Q13547 2/20 0.50
THRA P10827 2/20 0.50
THRB P10828 2/20 0.50
NPC1 O15118 1/20 0.50
POLB P06746 1/20 0.50
RAB9A P51151 1/20 0.50
KMT2A Q03164 1/20 0.50
MCOLN3 Q8TDD5 1/20 0.50
CTDSP1 Q9GZU7 1/20 0.50
HDAC6 Q9UBN7 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28465310 0.96 TRPV1 (0.58) TRPV1PLK1HDAC8RARBPLK3
SCHEMBL28459351 0.91 PLK1 (0.61) TRPV1PLK1HDAC8TMEM97SIGMAR1
SCHEMBL28469389 0.85 PLK1 (0.59) TRPV1PLK1HDAC1NPC1POLB
SCHEMBL24534682 0.82 PLK1 (0.67) TRPV1PLK1RARBTHRATHRB
SCHEMBL28466232 0.82 PLK1 (0.57) TRPV1PLK1RARBTHRATHRB
SCHEMBL28462599 0.82 MEN1 (0.60) PLK1NPC1POLBRAB9AKMT2A
SCHEMBL28463607 0.80 NR1H4 (0.59) PLK1RARBNPC1POLBRAB9A
SCHEMBL6551314 0.79 ALDH1A1 (0.55) HDAC8HDAC1NPC1RAB9AKMT2A
SCHEMBL7638853 0.79 TRPV1 (0.65) TRPV1PLK1RARBTHRATHRB
SCHEMBL22505170 0.78 PLK1 (0.65) TRPV1PLK1RARBTHRATHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111747904-A Polyfluoroalkenyl substituted oxazole compound and preparation method thereof 南京工业大学 2020-10-09 CN claimed
CN-111747904-A Polyfluoroalkenyl substituted oxazole compound and preparation method thereof 南京工业大学 2020-10-09 CN disclosed