SCHEMBL28469503

SCHEMBL28469503

O=C(O)OCC=Cc1ccc(C(F)(F)F)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.53
GRIK1 P39086 1/20 0.50
GRIK2 Q13002 1/20 0.50
HDAC3 O15379 1/20 0.49
ADAM17 P78536 1/20 0.49
HDAC1 Q13547 1/20 0.49
HDAC2 Q92769 1/20 0.49
HDAC10 Q969S8 1/20 0.49
HDAC11 Q96DB2 1/20 0.49
HDAC8 Q9BY41 1/20 0.49
HDAC6 Q9UBN7 1/20 0.49
HDAC5 Q9UQL6 1/20 0.49
PTGS1 P23219 1/20 0.47
PPARA Q07869 1/20 0.46
CYP1A1 P04798 5/20 0.45
CYP1B1 Q16678 5/20 0.45
MAOB P27338 3/20 0.45
CA1 P00915 1/20 0.45
CA2 P00918 1/20 0.45
S1PR5 Q9H228 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28469501 0.89 CYP1A2 (0.54) CYP1A2GRIK1GRIK2HDAC3ADAM17
SCHEMBL28849820 0.83 NOS3 (0.52) CYP1A2GRIK1GRIK2HDAC3ADAM17
SCHEMBL28469492 0.81 HSD11B1 (0.48) CYP1A2GRIK1GRIK2PTGS1MAOB
SCHEMBL6080800 0.80 CYP1A2 (0.45) CYP1A2GRIK1GRIK2HDAC3ADAM17
SCHEMBL6080803 0.80 CYP1A2 (0.45) CYP1A2GRIK1GRIK2HDAC3ADAM17
SCHEMBL3324115 0.79 IDO1 (0.57) CYP1A2HDAC3HDAC1HDAC2HDAC10
SCHEMBL293068 0.79 IDO1 (0.57) CYP1A2HDAC3HDAC1HDAC2HDAC10
SCHEMBL28469057 0.78 RAB9A (0.47) GRIK1GRIK2PPARACYP1B1MAOB
SCHEMBL28476052 0.78 CYP1A2 (0.48) CYP1A2GRIK1GRIK2HDAC3HDAC1
SCHEMBL28462213 0.78 GRIK1 (0.48) CYP1A2GRIK1GRIK2CYP1B1MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106316813-B 3-substituted 3-vinyl-2-hydroxy-1-aryl acetone and synthesis method thereof 上海交通大学 2020-09-15 CN disclosed