SCHEMBL28472385

SCHEMBL28472385

COC(=O)c1ccccc1N1C(=O)C=CC1=O

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TLR9 Q9NR96 2/20 0.58
ALDH1A1 P00352 2/20 0.58
ATM Q13315 2/20 0.58
MYC P01106 1/20 0.58
HSP90AA1 P07900 1/20 0.58
PKM P14618 1/20 0.58
CCR6 P51684 1/20 0.58
NPSR1 Q6W5P4 1/20 0.58
TDP1 Q9NUW8 1/20 0.58
SMN1; SMN2 Q16637 1/20 0.57
POLB P06746 2/20 0.55
MEN1 O00255 2/20 0.55
KMT2A Q03164 2/20 0.55
MGLL Q99685 8/20 0.54
TSHR P16473 3/20 0.50
LMNA P02545 1/20 0.50
CFTR P13569 1/20 0.49
HSD17B10 Q99714 1/20 0.49
KDM4E B2RXH2 2/20 0.47
FAAH O00519 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15434915 0.85 MYC (0.66) ALDH1A1ATMMYCSMN1; SMN2POLB
SCHEMBL15033486 0.82 TSHR (0.61) TLR9ALDH1A1ATMHSP90AA1PKM
SCHEMBL11357026 0.81 TDP1 (0.57) TLR9ALDH1A1ATMHSP90AA1PKM
SCHEMBL29510541 0.80 TLR9 (0.64) TLR9ALDH1A1ATMMYCHSP90AA1
SCHEMBL9240798 0.80 TLR9 (0.64) TLR9ALDH1A1ATMMYCHSP90AA1
SCHEMBL15129225 0.80 ALDH1A1 (0.59) TLR9ALDH1A1ATMHSP90AA1PKM
SCHEMBL28752508 0.79 TLR9 (0.63) TLR9ALDH1A1ATMHSP90AA1PKM
SCHEMBL18470139 0.79 MYC (0.54) ALDH1A1ATMMYCSMN1; SMN2POLB
SCHEMBL29364136 0.78 ALDH1A1 (0.71) TLR9ALDH1A1ATMMYCHSP90AA1
SCHEMBL183052 0.78 ALDH1A1 (0.71) TLR9ALDH1A1ATMMYCHSP90AA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114432301-B Covalent inhibitor derivative and application thereof in treatment of viral infection 北京大学 2024-05-31 CN disclosed
CN-114432301-A Covalent inhibitor derivative and application thereof in treating virus infection 北京大学 2022-05-06 CN disclosed
CN-109180553-B Preparation method of p53 allosteric preparation and application of allosteric preparation as medicine 中国药科大学 2020-10-16 CN disclosed