SCHEMBL28475487

SCHEMBL28475487

COc1ccc(-c2cc3c(cn2)[nH]c(=O)n3-c2cc(OC)c(OC)c(OC)c2)cc1C(=O)O

nearest known ligand 0.51

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
KATNA1 O75449 1/20 0.51
MAP3K11 Q16584 13/20 0.43
LRRK2 Q5S007 1/20 0.40
NEK2 P51955 4/20 0.40
TP53 P04637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29176281 0.87 KATNA1 (0.64) KATNA1MAP3K11LRRK2
SCHEMBL30800023 0.87 KATNA1 (0.64) KATNA1MAP3K11LRRK2
SCHEMBL30800088 0.86 KATNA1 (0.47) KATNA1MAP3K11LRRK2
SCHEMBL29176307 0.86 KATNA1 (0.47) KATNA1MAP3K11LRRK2
SCHEMBL29176285 0.86 KATNA1 (0.50) KATNA1MAP3K11LRRK2
SCHEMBL29176283 0.85 KATNA1 (0.52) KATNA1MAP3K11LRRK2
SCHEMBL30799989 0.85 KATNA1 (0.52) KATNA1MAP3K11LRRK2
SCHEMBL28469098 0.84 MAP3K11 (0.53) KATNA1MAP3K11LRRK2
SCHEMBL29176290 0.83 KATNA1 (0.46) KATNA1MAP3K11LRRK2TP53
SCHEMBL29176294 0.82 KATNA1 (0.47) KATNA1MAP3K11LRRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111732584-B Diaryl substituted fused heterocycle compound and preparation method and application thereof in pharmacy 复旦大学 2024-02-27 CN disclosed
CN-111732584-A Diaryl substituted fused heterocyclic compound, preparation method thereof and application thereof in pharmacy 复旦大学 2020-10-02 CN disclosed