SCHEMBL28477707

SCHEMBL28477707

CC1(C)CCN(CCCBr)CC1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.36
DRD3 P35462 1/20 0.36
S1PR1 P21453 1/20 0.33
S1PR3 Q99500 1/20 0.33
S1PR5 Q9H228 1/20 0.33
HRH3 Q9Y5N1 1/20 0.32
CYP1A2 P05177 1/20 0.31
CYP2D6 P10635 1/20 0.31
ALOX15 P16050 1/20 0.31
NOS3 P29474 1/20 0.30
NOS1 P29475 1/20 0.30
NOS2 P35228 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21246950 0.83 S1PR1 (0.38) DRD2S1PR1S1PR3S1PR5HRH3
SCHEMBL21246968 0.83 NOS3 (0.32) S1PR1S1PR3S1PR5HRH3NOS3
SCHEMBL18091474 0.79 HRH3 (0.44) S1PR1S1PR3S1PR5HRH3NOS3
SCHEMBL18506727 0.79 S1PR1 (0.49) DRD2DRD3S1PR1S1PR3S1PR5
SCHEMBL24683346 0.77 DRD2 (0.36) DRD2DRD3S1PR1S1PR3S1PR5
SCHEMBL25355767 0.77 DRD2 (0.36) DRD2DRD3S1PR1S1PR3S1PR5
SCHEMBL24179174 0.77 S1PR1 (0.51) S1PR1S1PR3S1PR5
SCHEMBL2209695 0.77 KEAP1 (0.50) DRD2DRD3CYP2D6ALOX15
SCHEMBL23226782 0.77 HRH3 (0.33) HRH3NOS3NOS1NOS2
Bromide SCHEMBL20551357 0.77 HRH3 (0.42) HRH3NOS3NOS1NOS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111788207-B Dioxane quinoline compound and preparation method and application thereof 北京赛特明强医药科技有限公司 2021-03-23 CN disclosed
CN-111788207-A Dioxane quinoline compound and preparation method and application thereof 北京赛特明强医药科技有限公司 2020-10-16 CN disclosed