SCHEMBL28478702

SCHEMBL28478702

O=C(c1ccc(Cl)cn1)N1CC[CH]CC1

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.48
GRM5 P41594 2/20 0.45
HRH3 Q9Y5N1 1/20 0.44
PRKAA2 P54646 2/20 0.44
PRKAB2 O43741 1/20 0.44
PRKAG1 P54619 1/20 0.44
PRKAA1 Q13131 1/20 0.44
PRKAG3 Q9UGI9 1/20 0.44
PRKAG2 Q9UGJ0 1/20 0.44
PRKAB1 Q9Y478 1/20 0.44
L3MBTL1 Q9Y468 2/20 0.44
L3MBTL3 Q96JM7 1/20 0.43
MAOB P27338 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
AOC3 Q16853 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1507073 0.85 GRM5 (0.59) SMN1; SMN2GRM5HRH3L3MBTL1L3MBTL3
SCHEMBL1809378 0.75 HRH3 (0.54) HRH3PRKAA2PRKAB2PRKAG1PRKAA1
SCHEMBL979538 0.74 ALDH1A1 (0.66) RAB9A
SCHEMBL9792343 0.73 L3MBTL1 (0.80) SMN1; SMN2L3MBTL1
SCHEMBL28477730 0.71 RAB9A (0.62) SMN1; SMN2GRM5PRKAA2PRKAB2PRKAG1
SCHEMBL28467301 0.71 GNE (0.51) SMN1; SMN2GRM5L3MBTL1NPC1RAB9A
SCHEMBL10815017 0.70 MAOB (0.55) SMN1; SMN2L3MBTL1MAOBTDP1NPC1
SCHEMBL28254880 0.70 CYP3A4 (0.56)
SCHEMBL1441384 0.69 MAOB (0.53) SMN1; SMN2L3MBTL1MAOBTDP1NPC1
SCHEMBL211889 0.69 P4HTM (0.59) L3MBTL1MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112370452-A Heterocyclic amides as kinase inhibitors 葛兰素史密斯克莱知识产权发展有限公司 2021-02-19 CN disclosed
CN-107624111-B Heterocyclic amides as kinase inhibitors 葛兰素史密斯克莱知识产权发展有限公司 2020-11-03 CN disclosed