SCHEMBL28479219

SCHEMBL28479219

CC1(Nc2ccc(C(N)=O)nn2)COC1

nearest known ligand 0.41

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
NNMT P40261 2/20 0.41
GSK3B P49841 1/20 0.34
KIF18A Q8NI77 3/20 0.34
CYP1A2 P05177 1/20 0.33
GABRA1 P14867 3/20 0.31
BACE1 P56817 2/20 0.30
BACE2 Q9Y5Z0 2/20 0.30
CNR2 P34972 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28474245 0.86 NNMT (0.45) NNMTGSK3B
SCHEMBL28473395 0.72 NNMT (0.42) NNMTGSK3BBACE1
Hydracarbazine SCHEMBL308554 0.70 NNMT (0.55) NNMTGSK3B
SCHEMBL4889620 0.69 HCAR3 (0.46) NNMT
SCHEMBL3174330 0.69 NNMT (0.67) NNMTGSK3B
SCHEMBL7667785 0.68 NNMT (0.49) NNMTGSK3B
SCHEMBL28479050 0.68 GSK3B (0.50) NNMTGSK3B
SCHEMBL31211632 0.67 NNMT (0.47) NNMTGSK3B
SCHEMBL30542994 0.67 NNMT (0.44) NNMTGSK3BKIF18AGABRA1CNR2
SCHEMBL28477862 0.65 GSK3B (0.44) NNMTGSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115448910-A Pyridazine derivative inhibitor, and preparation method and application thereof 江苏豪森药业集团有限公司 2022-12-09 CN disclosed
CN-111757878-A Pyridazine derivative inhibitor, and preparation method and application thereof 江苏豪森药业集团有限公司 2020-10-09 CN disclosed