SCHEMBL284797

SCHEMBL284797

C=COC(=O)OCCOC(=O)OC=C

nearest known ligand 0.42

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TSHR P16473 6/20 0.42
ALDH1A1 P00352 3/20 0.42
TP53 P04637 2/20 0.42
HIF1A Q16665 2/20 0.42
HSD17B10 Q99714 1/20 0.42
CYP3A4 P08684 1/20 0.37
HPGD P15428 1/20 0.33
THRB P10828 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL284310 0.93 TSHR (0.54) TSHRALDH1A1TP53HIF1AHSD17B10
SCHEMBL1799910 0.90 TSHR (0.44) TSHRALDH1A1TP53HIF1AHSD17B10
SCHEMBL284885 0.90 TSHR (0.50) TSHRALDH1A1TP53HIF1AHSD17B10
SCHEMBL8004719 0.89 TSHR (0.35) TSHRALDH1A1TP53HIF1AHSD17B10
SCHEMBL12607040 0.89 TSHR (0.61) TSHRALDH1A1TP53HIF1AHSD17B10
SCHEMBL11332982 0.87 CA2 (0.37) TSHRALDH1A1TP53HIF1AHSD17B10
SCHEMBL284174 0.87 TSHR (0.54) TSHRALDH1A1TP53HIF1AHSD17B10
SCHEMBL35344 0.87
SCHEMBL13248945 0.87 ALDH1A1 (0.54) TSHRALDH1A1TP53HIF1AHSD17B10
SCHEMBL167897 0.85

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 73 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117425984-A Flame-resistant electrode for lithium battery comprising quasi-solid electrolyte or solid electrolyte and method of manufacture 环球石墨烯集团公司 2024-01-19 CN claimed
CN-117321804-A Bipolar electrode comprising a flame-resistant quasi-solid electrolyte or solid electrolyte, bipolar lithium battery and method for producing same 环球石墨烯集团公司 2023-12-29 CN claimed
CN-117321807-A Flame-retardant bipolar electrode, bipolar lithium battery and manufacturing method 环球石墨烯集团公司 2023-12-29 CN claimed
CN-117044003-A Flame-retardant quasi-solid electrolyte, lithium battery and manufacturing method 环球石墨烯集团公司 2023-11-10 CN claimed
CN-115719828-A Rechargeable lithium battery 三星SDI株式会社 2023-02-28 CN claimed
US-10668676-B2 Ophthalmic devices BAUSCH & LOMB INCORPORATED (US) 2020-06-02 US claimed
US-20200047437-A1 OPHTHALMIC DEVICES MEDICIS PHARMACEUTICAL CORPORATION 2020-02-13 US claimed
EP-3091050-B1 THIOL-ENE POLYMERIZATION WITH VINYLESTERS AND VINYLCARBONATE SYNTHES GMBH (CH) 2018-07-18 EP claimed
US-9814801-B2 Thiol-ene polymerization with vinylesters and vinylcarbonate DePuy Synthes Products, Inc. (US) 2017-11-14 US claimed
EP-3091050-A1 THIOL-ENE POLYMERIZATION WITH VINYLESTERS AND VINYLCARBONATE Synthes GmbH (CH) 2016-11-09 EP claimed
US-20160243279-A1 THIOL-ENE POLYMERIZATION WITH VINYLESTERS AND VINYLCARBONATE SYNTHES GMBH (CH) 2016-08-25 US claimed
EP-2764049-B1 THIOL-ENE POLYMERIZATION WITH VINYLESTERS AND VINYLCARBONATE SYNTHES GMBH (CH) 2016-08-17 EP claimed
EP-2764049-A1 THIOL-ENE POLYMERIZATION WITH VINYLESTERS AND VINYLCARBONATE Synthes GmbH (CH) 2014-08-13 EP claimed
WO-2013052328-A1 THIOL-ENE POLYMERIZATION WITH VINYLESTERS AND VINYLCARBONATE SYNTHES USA, LLC (US) 2013-04-11 WO claimed
US-20130084543-A1 THIOL-ENE POLYMERIZATION WITH VINYLESTERS AND VINYLCARBONATE TECHNISCHE UNIVERSITAT WIEN (AT) 2013-04-04 US claimed
US-6166236-A Vinyl carbonate and vinyl carbamate contact lens material monomers BAUSCH & LOMB INCORPORATED (US) 2000-12-26 US claimed
EP-0396364-B1 Copolymers of vinyl carbonate and vinyl carbamate as contact lens material BAUSCH & LOMB (US) 1997-06-11 EP claimed
US-5610252-A Vinyl carbonate and vinyl carbamate contact lens material monomers BAUSCH & LOMB INCORPORATED (US) 1997-03-11 US claimed
EP-0396364-A2 Novel vinyl carbonate and vinyl carbamate contact lens material monomers BAUSCH & LOMB INCORPORATED (US) 1990-11-07 EP claimed
EP-4396616-A1 OPHTHALMIC DEVICES Bausch + Lomb Ireland Limited (IE) 2024-07-10 EP disclosed
US-11897985-B2 Water extractable ophthalmic devices BAUSCH & LOMB INCORPORATED (US) 2024-02-13 US disclosed
CN-117425984-A Flame-resistant electrode for lithium battery comprising quasi-solid electrolyte or solid electrolyte and method of manufacture 环球石墨烯集团公司 2024-01-19 CN disclosed
US-11873361-B2 Ophthalmic devices BAUSCH + LOMB IRELAND LIMITED (IE) 2024-01-16 US disclosed
CN-117321807-A Flame-retardant bipolar electrode, bipolar lithium battery and manufacturing method 环球石墨烯集团公司 2023-12-29 CN disclosed
CN-117321804-A Bipolar electrode comprising a flame-resistant quasi-solid electrolyte or solid electrolyte, bipolar lithium battery and method for producing same 环球石墨烯集团公司 2023-12-29 CN disclosed
CN-117044003-A Flame-retardant quasi-solid electrolyte, lithium battery and manufacturing method 环球石墨烯集团公司 2023-11-10 CN disclosed
US-20230089707-A1 OPHTHALMIC DEVICES JPMORGAN CHASE BANK, N.A., AS SUCCESSOR AGENT 2023-03-23 US disclosed
WO-2023030716-A1 OPHTHALMIC DEVICES BAUSCH + LOMB IRELAND LIMITED (IE) 2023-03-09 WO disclosed
US-11345773-B2 Water extractable ophthalmic devices BAUSCH & LOMB INCORPORATED (US) 2022-05-31 US disclosed
US-11022722-B2 Water extractable ophthalmic devices BAUSCH & LOMB INCORPORATED (US) 2021-06-01 US disclosed
US-10668676-B2 Ophthalmic devices BAUSCH & LOMB INCORPORATED (US) 2020-06-02 US disclosed
US-20200047437-A1 OPHTHALMIC DEVICES MEDICIS PHARMACEUTICAL CORPORATION 2020-02-13 US disclosed
US-20190352443-A1 WATER EXTRACTABLE OPHTHALMIC DEVICES BAUSCH HEALTH AMERICAS, INC. 2019-11-21 US disclosed
EP-3091050-B1 THIOL-ENE POLYMERIZATION WITH VINYLESTERS AND VINYLCARBONATE SYNTHES GMBH (CH) 2018-07-18 EP disclosed
US-9814801-B2 Thiol-ene polymerization with vinylesters and vinylcarbonate DePuy Synthes Products, Inc. (US) 2017-11-14 US disclosed
US-9814801-B2 Thiol-ene polymerization with vinylesters and vinylcarbonate DePuy Synthes Products, Inc. (US) 2017-11-14 US disclosed
US-9814801-B2 Thiol-ene polymerization with vinylesters and vinylcarbonate DePuy Synthes Products, Inc. (US) 2017-11-14 US disclosed
US-9623145-B2 Thiol-ene polymerization with vinylesters and vinylcarbonate DePuy Synthes Products, Inc. (US) 2017-04-18 US disclosed
US-9623145-B2 Thiol-ene polymerization with vinylesters and vinylcarbonate DePuy Synthes Products, Inc. (US) 2017-04-18 US disclosed
US-9623145-B2 Thiol-ene polymerization with vinylesters and vinylcarbonate DePuy Synthes Products, Inc. (US) 2017-04-18 US disclosed
EP-3091050-A1 THIOL-ENE POLYMERIZATION WITH VINYLESTERS AND VINYLCARBONATE Synthes GmbH (CH) 2016-11-09 EP disclosed
EP-3091050-A1 THIOL-ENE POLYMERIZATION WITH VINYLESTERS AND VINYLCARBONATE Synthes GmbH (CH) 2016-11-09 EP disclosed
US-20160243279-A1 THIOL-ENE POLYMERIZATION WITH VINYLESTERS AND VINYLCARBONATE SYNTHES GMBH (CH) 2016-08-25 US disclosed
US-20160243279-A1 THIOL-ENE POLYMERIZATION WITH VINYLESTERS AND VINYLCARBONATE SYNTHES GMBH (CH) 2016-08-25 US disclosed
US-20160243279-A1 THIOL-ENE POLYMERIZATION WITH VINYLESTERS AND VINYLCARBONATE SYNTHES GMBH (CH) 2016-08-25 US disclosed
EP-2764049-B1 THIOL-ENE POLYMERIZATION WITH VINYLESTERS AND VINYLCARBONATE SYNTHES GMBH (CH) 2016-08-17 EP disclosed
EP-2764049-B1 THIOL-ENE POLYMERIZATION WITH VINYLESTERS AND VINYLCARBONATE SYNTHES GMBH (CH) 2016-08-17 EP disclosed
US-8999323-B2 Composition that can be cured by polymerisation for the production of biodegradable, biocompatible, cross-linkable polymers on the basis of polyvinyl alcohol TECHNISCHE UNIVERSITÄT WIEN (AT) 2015-04-07 US disclosed
US-8999323-B2 Composition that can be cured by polymerisation for the production of biodegradable, biocompatible, cross-linkable polymers on the basis of polyvinyl alcohol TECHNISCHE UNIVERSITÄT WIEN (AT) 2015-04-07 US disclosed
US-8999323-B2 Composition that can be cured by polymerisation for the production of biodegradable, biocompatible, cross-linkable polymers on the basis of polyvinyl alcohol TECHNISCHE UNIVERSITÄT WIEN (AT) 2015-04-07 US disclosed
EP-2061115-B1 LITHIUM DIFLUOROPHOSPHATE, ELECTROLYTIC SOLUTION CONTAINING LITHIUM DIFLUOROPHOSPHATE, PROCESS FOR PRODUCING LITHIUM DIFLUOROPHOSPHATE, PROCESS FOR PRODUCING NONAQUEOUS ELECTROLYTIC SOLUTION, NONAQUEOUS ELECTROLYTIC SOLUTION, AND NONAQUEOUS-ELECTROLYTIC-SOLUTION SECONDARY CELL EMPLOYING THE SAME MITSUBISHI CHEM CORP (JP) 2015-04-01 EP disclosed
EP-2764049-A1 THIOL-ENE POLYMERIZATION WITH VINYLESTERS AND VINYLCARBONATE Synthes GmbH (CH) 2014-08-13 EP disclosed
EP-2428235-B1 Use of compounds hardened by means of polymerisation for producing biodegradable, biocompatible, networked polymers UNIV WIEN TECH (AT) 2014-06-04 EP disclosed
EP-2428235-B1 Use of compounds hardened by means of polymerisation for producing biodegradable, biocompatible, networked polymers UNIV WIEN TECH (AT) 2014-06-04 EP disclosed
WO-2013052328-A1 THIOL-ENE POLYMERIZATION WITH VINYLESTERS AND VINYLCARBONATE SYNTHES USA, LLC (US) 2013-04-11 WO disclosed
WO-2013052328-A1 THIOL-ENE POLYMERIZATION WITH VINYLESTERS AND VINYLCARBONATE SYNTHES USA, LLC (US) 2013-04-11 WO disclosed
US-20130084543-A1 THIOL-ENE POLYMERIZATION WITH VINYLESTERS AND VINYLCARBONATE TECHNISCHE UNIVERSITAT WIEN (AT) 2013-04-04 US disclosed
US-20130084543-A1 THIOL-ENE POLYMERIZATION WITH VINYLESTERS AND VINYLCARBONATE TECHNISCHE UNIVERSITAT WIEN (AT) 2013-04-04 US disclosed
US-20130084543-A1 THIOL-ENE POLYMERIZATION WITH VINYLESTERS AND VINYLCARBONATE TECHNISCHE UNIVERSITAT WIEN (AT) 2013-04-04 US disclosed
EP-2428235-A2 Use of compounds hardened by means of polymerisation for producing biodegradable, biocompatible, networked polymers Technische Universität Wien (AT) 2012-03-14 EP disclosed
EP-2428235-A2 Use of compounds hardened by means of polymerisation for producing biodegradable, biocompatible, networked polymers Technische Universität Wien (AT) 2012-03-14 EP disclosed
US-20100303804-A1 COMPOSITION THAT CAN BE CURED BY POLYMERISATION FOR THE PRODUCTION OF BIODEGRADABLE, BIOCOMPATIBLE, CROSS-LINKABLE POLYMERS ON THE BASIS OF POLYVINYL ALCOHOL TECHNISCHE UNIVERSITAT WIEN (AT) 2010-12-02 US disclosed
US-20100303804-A1 COMPOSITION THAT CAN BE CURED BY POLYMERISATION FOR THE PRODUCTION OF BIODEGRADABLE, BIOCOMPATIBLE, CROSS-LINKABLE POLYMERS ON THE BASIS OF POLYVINYL ALCOHOL TECHNISCHE UNIVERSITAT WIEN (AT) 2010-12-02 US disclosed
US-20100303804-A1 COMPOSITION THAT CAN BE CURED BY POLYMERISATION FOR THE PRODUCTION OF BIODEGRADABLE, BIOCOMPATIBLE, CROSS-LINKABLE POLYMERS ON THE BASIS OF POLYVINYL ALCOHOL TECHNISCHE UNIVERSITAT WIEN (AT) 2010-12-02 US disclosed
US-20090286155-A1 LITHIUM DIFLUOROPHOSPHATE, ELECTROLYTE CONTAINING LITHIUM DIFLUOROPHOSPHATE, PROCESS FOR PRODUCING LITHIUM DIFLUOROPHOSPHATE, PROCESS FOR PRODUCING NONAQUEOUS ELECTROLYTE, NONAQUEOUS ELECTROLYTE, AND NONAQUEOUS ELECTROLYTE SECONDARY BATTERY CONTAINING THE SAME MITSUBISHI CHEMICAL CORPORATION (JP) 2009-11-19 US disclosed
WO-2009065162-A2 COMPOSITION THAT CAN BE CURED BY POLYMERISATION FOR THE PRODUCTION OF BIODEGRADABLE, BIOCOMPATIBLE, CROSS-LINKABLE POLYMERS ON THE BASIS OF POLYVINYL ALCOHOL TECHNISCHE UNIVERSITÄT WIEN (AT) 2009-05-28 WO disclosed
EP-2061115-A1 LITHIUM DIFLUOROPHOSPHATE, ELECTROLYTIC SOLUTION CONTAINING LITHIUM DIFLUOROPHOSPHATE, PROCESS FOR PRODUCING LITHIUM DIFLUOROPHOSPHATE, PROCESS FOR PRODUCING NONAQUEOUS ELECTROLYTIC SOLUTION, NONAQUEOUS ELECTROLYTIC SOLUTION, AND NONAQUEOUS-ELECTROLYTIC-SOLUTION SECONDARY CELL EMPLOYING THE SAME Mitsubishi Chemical Corporation (JP) 2009-05-20 EP disclosed
US-6166236-A Vinyl carbonate and vinyl carbamate contact lens material monomers BAUSCH & LOMB INCORPORATED (US) 2000-12-26 US disclosed
EP-0396364-B1 Copolymers of vinyl carbonate and vinyl carbamate as contact lens material BAUSCH & LOMB (US) 1997-06-11 EP disclosed
US-5610252-A Vinyl carbonate and vinyl carbamate contact lens material monomers BAUSCH & LOMB INCORPORATED (US) 1997-03-11 US disclosed
EP-0757033-A2 Vinyl carbonate and vinyl carbamate monomers for a contact lens material BAUSCH & LOMB INCORPORATED (US) 1997-02-05 EP disclosed
US-5070215-A Gas permeable contact lenses BAUSCH & LOMB INCORPORATED (US) 1991-12-03 US disclosed
EP-0396364-A2 Novel vinyl carbonate and vinyl carbamate contact lens material monomers BAUSCH & LOMB INCORPORATED (US) 1990-11-07 EP disclosed
EP-0396364-A2 Novel vinyl carbonate and vinyl carbamate contact lens material monomers BAUSCH & LOMB INCORPORATED (US) 1990-11-07 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130084543-A1 THIOL-ENE POLYMERIZATION WITH VINYLESTERS AND VINYLCARBONATE TMT1A, MGMT, CBS TSHR 2137/4885ALDH1A1 335/4885TP53 2278/4885
US-20100303804-A1 COMPOSITION THAT CAN BE CURED BY POLYMERISATION FOR THE PRODUCTION OF BIODEGRADABLE, BIOCOMPATIBLE, CROSS-LINKABLE POLYMERS ON THE BASIS OF POLYVINYL ALCOHOL SCO2, CBR1, CBR3 TSHR 4555/4885ALDH1A1 822/4885TP53 3423/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.