SCHEMBL28484153

SCHEMBL28484153

NC(=O)c1cccc2c1nc(-c1ccc([N+](=O)[O-])cc1)n2Cc1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CFTR P13569 3/20 0.50
PARP1 P09874 4/20 0.49
AR P10275 6/20 0.48
PKN1 Q16512 1/20 0.48
PKN2 Q16513 1/20 0.48
PLA2G2A P14555 1/20 0.45
KMT2A Q03164 2/20 0.44
KDM4E B2RXH2 1/20 0.44
MITF O75030 1/20 0.44
MAPT P10636 1/20 0.44
HTT P42858 1/20 0.44
MEN1 O00255 1/20 0.43
POLB P06746 1/20 0.43
TBXA2R P21731 1/20 0.43
PDE6D O43924 1/20 0.43
ALDH1A1 P00352 1/20 0.43
ALDH2 P05091 1/20 0.43
ALDH3A1 P30838 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29412059 1.00 CFTR (0.50) CFTRPARP1ARPKN1PKN2
SCHEMBL28493353 0.90 CFTR (0.56) CFTRPARP1PKN1PKN2PLA2G2A
SCHEMBL29412022 0.90 CFTR (0.56) CFTRPARP1PKN1PKN2PLA2G2A
SCHEMBL28487665 0.88 PKN1 (0.56) PARP1PKN1PKN2MAPTPDE6D
SCHEMBL29412017 0.88 PKN1 (0.56) PARP1PKN1PKN2MAPTPDE6D
SCHEMBL28478408 0.86 ALDH1A1 (0.58) PARP1PKN1PKN2MAPTHTT
SCHEMBL29412060 0.86 PKN1 (0.54) PARP1PKN1PKN2KMT2AKDM4E
SCHEMBL28484147 0.85 PARP1 (0.51) PARP1PKN1PKN2KMT2AKDM4E
SCHEMBL29411964 0.85 PARP1 (0.51) PARP1PKN1PKN2KMT2AKDM4E
SCHEMBL29829700 0.84 CFTR (0.55) CFTRARMAPTHTTPDE6D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111978301-B Benzimidazole compound with endothelial lipase inhibition effect and application thereof 盐城师范学院 2022-08-02 CN disclosed
CN-111978301-A Benzimidazole compound with endothelial lipase inhibition effect and application thereof 盐城师范学院 2020-11-24 CN disclosed