SCHEMBL28484338

SCHEMBL28484338

O=C(NC1[CH]C1)c1cccc2ccn(Cc3ccc(-c4cnn(CCCO)c4)cn3)c12

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 1/20 0.34
MTOR P42345 1/20 0.34
ATM Q13315 1/20 0.34
ATR Q13535 1/20 0.34
HCRTR2 O43614 5/20 0.33
IKBKE Q14164 1/20 0.32
TBK1 Q9UHD2 1/20 0.32
NAMPT P43490 1/20 0.32
TYRO3 Q06418 1/20 0.32
MET P08581 1/20 0.31
KDR P35968 1/20 0.31
PTGER4 P35408 2/20 0.31
PTGDR Q13258 2/20 0.31
TBXA2R P21731 1/20 0.31
PTGER1 P34995 1/20 0.31
PTGFR P43088 1/20 0.31
PTGER3 P43115 1/20 0.31
PTGER2 P43116 1/20 0.31
MAPK1 P28482 2/20 0.31
PDK2 Q15119 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28485215 0.88 MERTK (0.38) MAPK1
SCHEMBL28494628 0.84 PTGER4 (0.37) PTGER4PTGDRTBXA2RPTGER1PTGFR
SCHEMBL28493538 0.82 CBLB (0.34) PTGER4PTGDRTBXA2RPTGER1PTGFR
SCHEMBL28480177 0.81 KCNH2 (0.36) PTGER4PTGDRTBXA2RPTGER1PTGFR
SCHEMBL22276148 0.81 TBXA2R (0.34) PIK3CAMTORATMATRHCRTR2
SCHEMBL23890360 0.81 TBXA2R (0.34) HCRTR2PTGER4PTGDRTBXA2RPTGER1
SCHEMBL22276183 0.80 TBXA2R (0.33) PIK3CAMTORATMATRPTGER4
SCHEMBL28492006 0.80 DNM1L (0.35) PTGER4PTGDRTBXA2RPTGER1PTGFR
SCHEMBL23890380 0.79 TBXA2R (0.33) PIK3CAMTORATMATRPTGER4
SCHEMBL28487314 0.77 PTGER4 (0.35) PTGER4PTGDRTBXA2RPTGER1PTGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111989311-B Compound for inhibiting PGE2/EP4 signal transduction, preparation method thereof and application thereof in medicines 凯复(苏州)生物医药有限公司 2022-03-22 CN disclosed
CN-111989311-A Compound for inhibiting PGE2/EP4 signal transduction, preparation method thereof and application thereof in medicines 凯复(苏州)生物医药有限公司 2020-11-24 CN disclosed