SCHEMBL28485993

SCHEMBL28485993

Cc1[c]c(S(=O)(=O)N2CCC(N)CC2)cc([N+](=O)[O-])c1

nearest known ligand 0.44

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.44
ALDH1A1 P00352 4/20 0.42
SMN1; SMN2 Q16637 3/20 0.42
MCOLN3 Q8TDD5 2/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
HTT P42858 1/20 0.39
RECQL P46063 1/20 0.39
EPHX2 P34913 2/20 0.37
MAPT P10636 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28472330 0.85 LMNA (0.43) LMNAALDH1A1SMN1; SMN2MCOLN3L3MBTL1
SCHEMBL28474493 0.83 HTT (0.47) ALDH1A1SMN1; SMN2L3MBTL1HTT
SCHEMBL28901016 0.81 L3MBTL1 (0.46) LMNAALDH1A1SMN1; SMN2MCOLN3L3MBTL1
SCHEMBL28474461 0.80 MAPT (0.56) LMNAALDH1A1SMN1; SMN2L3MBTL1HTT
SCHEMBL28480715 0.79 KMT2A (0.47) LMNAALDH1A1SMN1; SMN2L3MBTL1HTT
SCHEMBL28480755 0.79 ALDH1A1 (0.45) LMNAALDH1A1SMN1; SMN2MCOLN3L3MBTL1
SCHEMBL28480232 0.74 NPC1 (0.44) LMNAALDH1A1SMN1; SMN2HTTMAPT
SCHEMBL28473209 0.73 L3MBTL1 (0.37) LMNAALDH1A1SMN1; SMN2L3MBTL1HTT
SCHEMBL29202914 0.73 ALDH1A1 (0.40) LMNAALDH1A1SMN1; SMN2MCOLN3L3MBTL1
SCHEMBL14055643 0.73 SMN1; SMN2 (0.63) LMNAALDH1A1SMN1; SMN2HTTRECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111918864-A Prodrug compounds activated by AKR1C3 and their use to treat hyperproliferative disorders 阿基利斯医疗有限公司 2020-11-10 CN claimed
CN-111918864-A Prodrug compounds activated by AKR1C3 and their use to treat hyperproliferative disorders 阿基利斯医疗有限公司 2020-11-10 CN disclosed