SCHEMBL28486144

SCHEMBL28486144

OB(O)c1cc(Cl)ncc1C(F)(F)F

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3R1 P27986 1/20 0.37
PIK3CA P42336 1/20 0.37
ASPH Q12797 1/20 0.35
KCNQ3 O43525 2/20 0.34
KCNQ2 O43526 2/20 0.34
KCNE1 P15382 2/20 0.34
KCNQ1 P51787 2/20 0.34
AKR1C3 P42330 2/20 0.34
AKR1C2 P52895 2/20 0.34
JUN P05412 1/20 0.33
NFKB1 P19838 1/20 0.33
NFKB2 Q00653 1/20 0.33
RELA Q04206 1/20 0.33
PIK3CD O00329 1/20 0.32
COMT P21964 1/20 0.31
ALDH1A1 P00352 3/20 0.31
GAA P10253 1/20 0.31
HTT P42858 1/20 0.31
GPBAR1 Q8TDU6 1/20 0.31
CNR2 P34972 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29956331 0.79 ASPH (0.36) ASPH
SCHEMBL29953210 0.79 ASPH (0.36) ASPH
SCHEMBL29953406 0.78 PIK3CD (0.38) PIK3R1PIK3CAASPHAKR1C3PIK3CD
SCHEMBL2554225 0.76 CNR2 (0.32) CNR2
SCHEMBL3840400 0.76 PIK3R1 (0.42) PIK3R1PIK3CAASPHKCNQ3KCNQ2
SCHEMBL16115971 0.75 MEN1 (0.41) GAA
SCHEMBL29954959 0.75 KCNQ3 (0.33) KCNQ3KCNQ2KCNE1KCNQ1
SCHEMBL30503537 0.75 PIK3R1 (0.36) PIK3R1PIK3CAASPHKCNQ3KCNQ2
SCHEMBL432680 0.75 PIK3R1 (0.36) PIK3R1PIK3CAASPHKCNQ3KCNQ2
SCHEMBL29395367 0.75 PIK3R1 (0.36) PIK3R1PIK3CAASPHKCNQ3KCNQ2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111995587-A 1, 4-disubstituted 3, 4-dihydro-2 (3H) -quinazolinone compound and synthetic method and application thereof 上海工程技术大学 2020-11-27 CN claimed
US-20220340893-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2022-10-27 US disclosed
CN-111995587-B 1, 4-disubstituted 3, 4-dihydro-2 (3H) -quinazolinone compound and synthesis method and application thereof 上海工程技术大学 2022-10-21 CN disclosed
CN-111995587-A 1, 4-disubstituted 3, 4-dihydro-2 (3H) -quinazolinone compound and synthetic method and application thereof 上海工程技术大学 2020-11-27 CN disclosed