SCHEMBL28489283

SCHEMBL28489283

CC(C)(C)OC(=O)NC1CCN(c2ccc(C#N)c(Cl)c2)CC1

nearest known ligand 0.52

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
AR P10275 4/20 0.52
SUV39H2 Q9H5I1 7/20 0.51
CTSK P43235 2/20 0.47
KCNA3 P22001 1/20 0.47
RET P07949 1/20 0.46
DRD2 P14416 3/20 0.46
JAK3 P52333 1/20 0.45
BTK Q06187 1/20 0.45
CNR1 P21554 1/20 0.45
CNR2 P34972 1/20 0.45
DRD3 P35462 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13651242 0.94 SUV39H2 (0.57) ARSUV39H2CTSKDRD2JAK3
SCHEMBL5220499 0.87 KDM4D (0.53) ARSUV39H2CTSKKCNA3RET
SCHEMBL27655935 0.87 SUV39H2 (0.54) SUV39H2DRD2CNR1CNR2DRD3
SCHEMBL24508096 0.85 AR (0.51) ARSUV39H2CTSKKCNA3RET
SCHEMBL29663762 0.85 AR (0.51) ARSUV39H2CTSKKCNA3RET
SCHEMBL22557377 0.83 AR (0.60) AR
SCHEMBL5202966 0.82 CTSK (0.53) SUV39H2CTSKKCNA3RETDRD2
SCHEMBL25453973 0.82 SUV39H2 (0.50) SUV39H2DRD2CNR1CNR2DRD3
SCHEMBL12835697 0.82 SUV39H2 (0.54) SUV39H2CTSKKCNA3RETJAK3
SCHEMBL21397261 0.81 SUV39H2 (0.51) SUV39H2DRD2CNR1CNR2DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111825657-A Dual-function chimeric heterocyclic compound for targeted degradation of androgen receptor and application thereof 成都海创药业有限公司 2020-10-27 CN disclosed