SCHEMBL28490456

SCHEMBL28490456

O=C(O)N1CCN(c2cccc3c2cc(C(F)(F)F)n3Cc2ccsc2)CC1

nearest known ligand 0.37

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.36
HTR1A P08908 1/20 0.35
CCR2 P41597 1/20 0.33
IRAK4 Q9NWZ3 1/20 0.33
CETP P11597 1/20 0.33
GOT1 P17174 2/20 0.33
SIGMAR1 Q99720 1/20 0.33
CHRM2 P08172 1/20 0.33
CHRM1 P11229 1/20 0.33
CHRM3 P20309 1/20 0.33
NPC1 O15118 1/20 0.33
THRB P10828 1/20 0.33
GAA P10253 1/20 0.32
HTR6 P50406 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21302005 0.88 TP53 (0.39) ALDH1A1CHRM2CHRM1CHRM3
SCHEMBL30516347 0.87 ALDH1A1 (0.42) ALDH1A1HTR1ACETPHTR6
SCHEMBL21291583 0.87 ALDH1A1 (0.42) ALDH1A1HTR1ACETPHTR6
SCHEMBL21291606 0.84 HTR6 (0.41) ALDH1A1HTR1ASIGMAR1THRBHTR6
SCHEMBL30516342 0.84 HTR6 (0.41) ALDH1A1HTR1ASIGMAR1THRBHTR6
SCHEMBL28502343 0.83 CCR2 (0.38) ALDH1A1CCR2SIGMAR1
SCHEMBL30516380 0.83 PLA2G1B (0.45) ALDH1A1CCR2HTR6
SCHEMBL28509589 0.83 DRD4 (0.39) ALDH1A1THRB
Hydrochloric Acid SCHEMBL30516392 0.83 HTR6 (0.40) ALDH1A1HTR1ASIGMAR1THRBHTR6
SCHEMBL30516369 0.82 SRPK1 (0.43) ALDH1A1THRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112041300-A Indole and benzimidazole derivatives as dual 5-HT2A and5-HT 6receptor antagonists 阿达梅德制药公司 2020-12-04 CN disclosed