SCHEMBL28490668

SCHEMBL28490668

COc1cc(NC(=O)Nc2cc(Nc3ccc(C(C)(C)C)cc3)ncn2)cc(OC)c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 7/20 0.60
FGFR1 P11362 2/20 0.60
ERBB3 P21860 5/20 0.56
NPC1 O15118 4/20 0.55
RAB9A P51151 4/20 0.55
MAPT P10636 2/20 0.55
MAPK1 P28482 2/20 0.55
HTT P42858 2/20 0.55
SMN1; SMN2 Q16637 2/20 0.55
LMNA P02545 1/20 0.55
STAT1 P42224 1/20 0.55
MEN1 O00255 5/20 0.52
KMT2A Q03164 5/20 0.52
FGFR3 P22607 3/20 0.49
RAF1 P04049 1/20 0.47
BRAF P15056 1/20 0.47
TUBB4A P04350 1/20 0.47
TUBB P07437 1/20 0.47
TUBA3C P0DPH7 1/20 0.47
TUBA1B P68363 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28903919 0.80 EGFR (0.55) EGFRFGFR1ERBB3RAF1BRAF
SCHEMBL374439 0.80 EGFR (0.72) EGFRFGFR1ERBB3NPC1RAB9A
SCHEMBL374158 0.79 FGFR3 (0.77) EGFRFGFR1ERBB3FGFR3
SCHEMBL28495163 0.76 EGFR (0.58) EGFRFGFR1ERBB3NPC1RAB9A
SCHEMBL28261624 0.75 EGFR (1.00) EGFRFGFR1ERBB3NPC1RAB9A
SCHEMBL28498357 0.75 EGFR (0.66) EGFRFGFR1ERBB3NPC1RAB9A
SCHEMBL5814747 0.74 MAPK10 (0.61) EGFRFGFR1ERBB3NPC1RAB9A
SCHEMBL374665 0.73 FGFR3 (0.64) EGFRFGFR1ERBB3NPC1RAB9A
SCHEMBL373717 0.73 EGFR (0.80) EGFRFGFR1ERBB3NPC1RAB9A
SCHEMBL5752852 0.72 MEN1 (0.62) NPC1RAB9AMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109053594-B 1- (3, 5-dimethoxyphenyl) -3- (substituted pyrimidine-4-yl) urea compound and preparation and application thereof 温州医科大学 2020-12-18 CN disclosed