SCHEMBL2849786

SCHEMBL2849786

CC[C@@]12CCC[C@H]1[C@@H]1CCc3cc(NS(=O)(=O)O)c(OC)cc3[C@H]1CC2

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B1 P14061 3/20 0.48
ESR1 P03372 2/20 0.48
CYP19A1 P11511 2/20 0.47
STS P08842 10/20 0.46
CA2 P00918 4/20 0.46
CA9 Q16790 3/20 0.45
CYP1A2 P05177 2/20 0.43
CYP3A4 P08684 2/20 0.43
HSD17B10 Q99714 2/20 0.43
CYP1A1 P04798 2/20 0.43
CYP1B1 Q16678 2/20 0.43
LMNA P02545 2/20 0.43
MAPT P10636 2/20 0.43
TP53 P04637 1/20 0.43
TSHR P16473 1/20 0.43
NFKB1 P19838 1/20 0.43
CYP2C19 P33261 1/20 0.43
THPO P40225 1/20 0.43
MEN1 O00255 1/20 0.43
GMNN O75496 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2854229 0.84 CA2 (0.49) HSD17B1ESR1CYP19A1STSCA2
SCHEMBL2856714 0.83 ESR1 (0.64) HSD17B1ESR1CYP19A1CA2CA9
SCHEMBL2855545 0.82 STS (0.52) HSD17B1ESR1CYP19A1STSCA2
SCHEMBL2858825 0.82 STS (0.52) HSD17B1ESR1CYP19A1STSCA2
SCHEMBL2849377 0.82 STS (0.66) STSCA2CA9
SCHEMBL2849680 0.82 STS (0.47) HSD17B1ESR1CYP19A1STSCA2
SCHEMBL2853440 0.81 HSD17B1 (0.46) HSD17B1ESR1CYP19A1STSCA2
SCHEMBL3383953 0.81 ESR1 (0.49) HSD17B1ESR1CYP19A1STSCA2
SCHEMBL3379141 0.81 CA2 (0.63) HSD17B1ESR1CYP19A1STSCA2
SCHEMBL3379139 0.81 CA2 (0.63) HSD17B1ESR1CYP19A1STSCA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1594884-B1 ANTITUMORAL 18A-HOMOESTRA-1,3,5(10)-TRIEN-3-YL 2-SUBSTITUTED SULFAMATES STERIX LTD (GB) 2010-01-13 EP claimed