SCHEMBL28501475

SCHEMBL28501475

CC(Nc1ccnc2ccccc12)c1ccc([N+](=O)[O-])cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CRHBP P24387 1/20 0.50
CRHR2 Q13324 1/20 0.50
TAAR1 Q96RJ0 1/20 0.47
ALDH1A1 P00352 4/20 0.47
HTT P42858 3/20 0.47
GAA P10253 1/20 0.47
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
HIF1A Q16665 1/20 0.46
HSD17B10 Q99714 1/20 0.46
KMT2A Q03164 3/20 0.44
POLB P06746 1/20 0.44
CCNC P24863 1/20 0.44
CDK8 P49336 1/20 0.44
GALR3 O60755 1/20 0.42
NR2F2 P24468 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30307409 0.82 GALR3 (0.59) TAAR1ALDH1A1HTTKMT2AGALR3
SCHEMBL28511396 0.81 KMT2A (0.67) CRHBPCRHR2ALDH1A1HTTGAA
SCHEMBL28509057 0.80 GALR3 (0.69) CRHBPCRHR2ALDH1A1HTTGAA
SCHEMBL28220542 0.80 GAA (0.53) TAAR1HTTGAAGALR3NR2F2
SCHEMBL28506233 0.80 CRHBP (0.53) CRHBPCRHR2ALDH1A1HTTGAA
SCHEMBL15094547 0.78 KMT2A (0.62) HTTKMT2APOLBMEN1KDM4E
SCHEMBL28500108 0.78 ALDH1A1 (0.50) CRHBPCRHR2ALDH1A1HTTGAA
SCHEMBL28499026 0.77 IGF1R (0.61) CRHBPCRHR2ALDH1A1HTTGAA
SCHEMBL28501477 0.75 CRHBP (0.50) CRHBPCRHR2ALDH1A1HTTGAA
SCHEMBL8783600 0.74 ALDH1A1 (0.57) ALDH1A1HTTKMT2AGALR3NR2F2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112204010-B Heterocyclic derivatives and uses thereof C&C新药研究所 2024-03-19 CN claimed
CN-112204010-A Heterocyclic derivatives and use thereof C&C新药研究所 2021-01-08 CN claimed
CN-112204010-B Heterocyclic derivatives and uses thereof C&C新药研究所 2024-03-19 CN disclosed
CN-112204010-A Heterocyclic derivatives and use thereof C&C新药研究所 2021-01-08 CN disclosed