SCHEMBL28502016

SCHEMBL28502016

O=Cc1ccnc2ccc(-c3ccc(N4CCOCC4)cc3)cc12

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPKAPK2 P49137 8/20 0.57
MAPK10 P53779 1/20 0.53
PIK3CD O00329 2/20 0.52
PIK3CA P42336 2/20 0.52
PIK3CB P42338 2/20 0.52
PIK3CG P48736 1/20 0.52
PRKDC P78527 1/20 0.52
ACVR1B P36896 2/20 0.52
TGFBR1 P36897 2/20 0.52
BMPR1B O00238 1/20 0.52
PDGFRB P09619 1/20 0.52
KIT P10721 1/20 0.52
PDGFRA P16234 1/20 0.52
BMPR1A P36894 1/20 0.52
ACVRL1 P37023 1/20 0.52
ACVR1 Q04771 1/20 0.52
LMNA P02545 3/20 0.46
ALDH1A1 P00352 2/20 0.46
CYP3A4 P08684 2/20 0.46
MAPK1 P28482 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28502019 0.82 ACVR1 (0.50) MAPKAPK2PIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL28505160 0.82 MAPKAPK2 (0.60) MAPKAPK2MAPK10PIK3CDPIK3CAPIK3CB
SCHEMBL20732829 0.82 MAPKAPK2 (0.60) MAPKAPK2MAPK10PIK3CDPIK3CAPIK3CB
SCHEMBL31464797 0.82 MAPKAPK2 (0.66) MAPKAPK2MAPK10PRKDCACVR1BTGFBR1
SCHEMBL20733053 0.81 MAPKAPK2 (0.56) MAPKAPK2MAPK10ACVR1BTGFBR1BMPR1B
SCHEMBL20732831 0.80 MAPKAPK2 (0.55) MAPKAPK2MAPK10PIK3CAACVR1BTGFBR1
SCHEMBL20732830 0.78 MAPKAPK2 (0.53) MAPKAPK2MAPK10ACVR1BTGFBR1BMPR1B
SCHEMBL24532577 0.78 IP6K1 (0.54) MAPKAPK2PIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL8681101 0.76 PIK3CA (0.56) MAPKAPK2MAPK10PIK3CAACVR1
SCHEMBL20732922 0.76 MAPKAPK2 (0.53) MAPKAPK2MAPK10ACVR1BTGFBR1BMPR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111670183-A Novel heterocyclic compounds as CDK8/19 inhibitors BIOCAD股份公司 2020-09-15 CN claimed