SCHEMBL285059

SCHEMBL285059

CCCCCOC(=O)Nc1nc(=O)n([C@@H]2O[C@H](C)[C@@H](OC(C)=O)[C@H]2OC(C)=O)cc1F

nearest known ligand 0.75

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
LMNA P02545 4/20 0.75
ADK P55263 1/20 0.35
TDP1 Q9NUW8 2/20 0.33
THRB P10828 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
HIF1A Q16665 1/20 0.33
NAAA Q02083 2/20 0.31
HPGD P15428 1/20 0.31
RAB9A P51151 1/20 0.31
PKM P14618 1/20 0.31
ALDH1A1 P00352 2/20 0.31
TSHR P16473 1/20 0.31
TP53 P04637 1/20 0.30
MAPT P10636 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12302023 1.00 LMNA (0.75) LMNAADKTDP1THRBSMN1; SMN2
SCHEMBL12302015 1.00 LMNA (0.75) LMNAADKTDP1THRBSMN1; SMN2
SCHEMBL12945763 1.00 LMNA (0.75) LMNAADKTDP1THRBSMN1; SMN2
SCHEMBL12029798 1.00 LMNA (0.75) LMNAADKTDP1THRBSMN1; SMN2
SCHEMBL13340646 1.00 LMNA (0.75) LMNAADKTDP1THRBSMN1; SMN2
SCHEMBL8196421 1.00 LMNA (0.75) LMNAADKTDP1THRBSMN1; SMN2
SCHEMBL285464 0.99 LMNA (0.73) LMNAADKTDP1THRBSMN1; SMN2
SCHEMBL8992747 0.99 LMNA (0.73) LMNAADKTDP1THRBSMN1; SMN2
SCHEMBL16508681 0.99 LMNA (0.73) LMNAADKTDP1THRBSMN1; SMN2
SCHEMBL16508671 0.99 LMNA (0.73) LMNAADKTDP1THRBSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 30 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2428213-A1 STABILIZED CHLORITE SOLUTIONS IN COMBINATION WITH FLUOROPYRIMIDINES FOR USE IN CANCER TREATMENT Nuvo Research AG (CH) 2012-03-14 EP claimed
EP-2370414-A2 PREPARATION OF CAPECITABINE Dr. Reddy's Laboratories, Ltd. (IN) 2011-10-05 EP claimed
US-20110224422-A1 PREPARATION OF CAPECITABINE DR. REDDY'S LABORATORIES LTD. (IN) 2011-09-15 US claimed
EP-2241556-A1 METHOD FOR THE PREPARATION OF CAPECITABINE AND INTERMEDIATES USED IN SAID METHOD Coll Farma S.L. (ES) 2010-10-20 EP claimed
WO-2010065586-A2 PREPARATION OF CAPECITABINE DR. REDDY'S LABORATORIES LTD. (IN) 2010-06-10 WO claimed
EP-0882734-B1 5'-Deoxy-cytidine derivatives HOFFMANN LA ROCHE (CH) 2009-08-26 EP claimed
EP-1060183-B1 5'-DEOXYCYTIDINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2003-04-23 EP claimed
US-6211166-B1 COADMINISTERED WITH A 5-FLUOROURACIL DERIVATIVE; ANTICARCINOGENIC AGENTS HOFFMAN-LA ROCHE INC. 2001-04-03 US claimed
EP-0882734-A2 5'-Deoxy-cytidine derivatives F. HOFFMANN-LA ROCHE AG (CH) 1998-12-09 EP claimed
EP-0602454-B1 N-Oxycarbonyl substituted 5'-deoxy-5-fluorocytidines HOFFMANN LA ROCHE (CH) 1996-04-24 EP claimed
EP-0602454-A1 N-Oxycarbonyl substituted 5'-deoxy-5-fluorocytidines F. HOFFMANN-LA ROCHE AG (CH) 1994-06-22 EP claimed
CN-103601777-A Preparation method of capecitabine HARBIN PHARMACEUTICAL GROUP CO LTD GENERAL PHARMACEUTICAL FACTORY 2014-02-26 CN disclosed
EP-2428213-A1 STABILIZED CHLORITE SOLUTIONS IN COMBINATION WITH FLUOROPYRIMIDINES FOR USE IN CANCER TREATMENT Nuvo Research AG (CH) 2012-03-14 EP disclosed
EP-2370414-A2 PREPARATION OF CAPECITABINE Dr. Reddy's Laboratories, Ltd. (IN) 2011-10-05 EP disclosed
US-20110224422-A1 PREPARATION OF CAPECITABINE DR. REDDY'S LABORATORIES LTD. (IN) 2011-09-15 US disclosed
EP-1060183-B1 5'-DEOXYCYTIDINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2003-04-23 EP disclosed
US-6211166-B1 COADMINISTERED WITH A 5-FLUOROURACIL DERIVATIVE; ANTICARCINOGENIC AGENTS HOFFMAN-LA ROCHE INC. 2001-04-03 US disclosed
EP-0882734-A2 5'-Deoxy-cytidine derivatives F. HOFFMANN-LA ROCHE AG (CH) 1998-12-09 EP disclosed
EP-0602454-B1 N-Oxycarbonyl substituted 5'-deoxy-5-fluorocytidines HOFFMANN LA ROCHE (CH) 1996-04-24 EP disclosed
EP-0602454-A1 N-Oxycarbonyl substituted 5'-deoxy-5-fluorocytidines F. HOFFMANN-LA ROCHE AG (CH) 1994-06-22 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110224422-A1 PREPARATION OF CAPECITABINE DPYD, TYMP, DCTD LMNA 2368/4885ADK 1020/4885TDP1 206/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.