SCHEMBL28510306

SCHEMBL28510306

O=Cc1ccccc1COc1cccc(F)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 7/20 0.54
MAOA P21397 4/20 0.54
SLC6A2 P23975 2/20 0.50
SLC6A4 P31645 2/20 0.50
HTR1A P08908 1/20 0.50
SLC6A3 Q01959 1/20 0.50
NPC1 O15118 1/20 0.49
RAB9A P51151 1/20 0.49
DCPS Q96C86 1/20 0.47
DAO P14920 1/20 0.46
HTR6 P50406 1/20 0.44
MRGPRX4 Q96LA9 1/20 0.43
CCNB2 O95067 1/20 0.43
CDK1 P06493 1/20 0.43
CDK4 P11802 1/20 0.43
CCNB1 P14635 1/20 0.43
CCND1 P24385 1/20 0.43
CCNB3 Q8WWL7 1/20 0.43
NR4A2 P43354 1/20 0.43
FFAR1 O14842 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2293283 0.83 ALDH1A1 (0.46) MAOBMAOANR4A2FFAR1
SCHEMBL1200712 0.82 SMN1; SMN2 (0.50) MAOBMAOASLC6A2SLC6A4HTR1A
SCHEMBL1539549 0.82 MAOB (0.54) MAOBMAOANPC1RAB9ACCNB2
SCHEMBL7171456 0.82 NPC1 (0.49) MAOBMAOANPC1RAB9ADCPS
SCHEMBL13793927 0.80 SLC6A2 (0.53) MAOBMAOASLC6A2SLC6A4HTR1A
SCHEMBL28510243 0.80 RAB9A (0.42) MAOBMAOANPC1RAB9ACCNB2
SCHEMBL2292237 0.79 SOD1 (0.50) MAOBMAOANPC1RAB9ACCNB2
SCHEMBL2286460 0.78 SOD1 (0.51) MAOBMAOANPC1RAB9ACCNB2
SCHEMBL2292569 0.78 NPC1 (0.46) MAOBMAOANPC1RAB9ACCNB2
SCHEMBL2289832 0.78 ALDH1A1 (0.58) DCPSCDK4CCND1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107522654-B Novel alpha-aminoamide derivatives and medicinal use thereof 中国人民解放军军事医学科学院毒物药物研究所 2020-09-01 CN disclosed