SCHEMBL28512160

SCHEMBL28512160

Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)nc2)n1

nearest known ligand 0.68

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.68
ALDH1A1 P00352 1/20 0.68
CYP3A4 P08684 1/20 0.68
TDP1 Q9NUW8 1/20 0.68
GAA P10253 4/20 0.60
TSHR P16473 2/20 0.59
PKM P14618 3/20 0.53
KMT2A Q03164 3/20 0.53
MEN1 O00255 1/20 0.53
POLB P06746 1/20 0.53
HSD17B10 Q99714 1/20 0.53
MAPT P10636 2/20 0.52
CYP2C9 P11712 1/20 0.52
KDM4E B2RXH2 1/20 0.51
LMNA P02545 1/20 0.51
ADRA2B P18089 1/20 0.51
RXFP1 Q9HBX9 2/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Sulfamethazine SCHEMBL17256221 0.81 ALDH1A1 (1.00) SMN1; SMN2ALDH1A1CYP3A4TDP1GAA
Sulfamethazine SCHEMBL29918086 0.81 ALDH1A1 (1.00) SMN1; SMN2ALDH1A1CYP3A4TDP1GAA
Sulfamethazine SCHEMBL151305 0.81 ALDH1A1 (1.00) SMN1; SMN2ALDH1A1CYP3A4TDP1GAA
Sulfamethazine SCHEMBL3495558 0.80 ALDH1A1 (0.97) SMN1; SMN2ALDH1A1CYP3A4TDP1GAA
Sulfamethazine SCHEMBL1442165 0.80 ALDH1A1 (0.97) SMN1; SMN2ALDH1A1CYP3A4TDP1GAA
Sulfamethazine SCHEMBL28567572 0.80 ALDH1A1 (0.97) SMN1; SMN2ALDH1A1CYP3A4TDP1GAA
Sulfamethazine SCHEMBL28028309 0.79 ALDH1A1 (0.94) SMN1; SMN2ALDH1A1CYP3A4TDP1GAA
SCHEMBL12903578 0.78 SMN1; SMN2 (0.76) SMN1; SMN2ALDH1A1CYP3A4TDP1GAA
SCHEMBL3505117 0.78 SMN1; SMN2 (0.70) SMN1; SMN2ALDH1A1CYP3A4TDP1GAA
Sulfamethazine SCHEMBL11708760 0.78 ALDH1A1 (0.91) SMN1; SMN2ALDH1A1CYP3A4TDP1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112375081-B Pyrrole [2,3-d ] pyrimidine derivative with CDK4, 6 or 9 inhibiting activity and preparation method and application thereof 中国医学科学院医药生物技术研究所 2022-04-12 CN disclosed
CN-112375081-A Pyrrole [2,3-d ] pyrimidine derivative with CDK4, 6 or 9 inhibiting activity and preparation method and application thereof 中国医学科学院医药生物技术研究所 2021-02-19 CN disclosed