SCHEMBL28512403

SCHEMBL28512403

Fc1ccc(Oc2cc3cc[nH]c3cc2Br)c(F)c1

nearest known ligand 0.56

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 6/20 0.56
AHR P35869 4/20 0.47
EPAS1 Q99814 1/20 0.45
GPR84 Q9NQS5 1/20 0.45
CSNK2A1 P68400 1/20 0.41
SCN8A Q9UQD0 3/20 0.37
SCN10A Q9Y5Y9 3/20 0.37
CYP2A6 P11509 1/20 0.37
NR4A2 P43354 1/20 0.37
KDR P35968 1/20 0.36
HSPB1 P04792 1/20 0.36
BRD4 O60885 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28512935 0.87 GPR84 (0.46) TRPA1AHRGPR84CSNK2A1CYP2A6
SCHEMBL28505468 0.86 CSNK2A1 (0.45) TRPA1AHREPAS1GPR84CSNK2A1
SCHEMBL28511617 0.82 AHR (0.46) TRPA1AHRGPR84CSNK2A1SCN8A
SCHEMBL2443701 0.78 AXL (0.48) TRPA1EPAS1CSNK2A1BRD4
SCHEMBL30194137 0.78 AXL (0.48) TRPA1EPAS1CSNK2A1BRD4
SCHEMBL28520341 0.77 TRPA1 (0.54) TRPA1
SCHEMBL916587 0.76 GPR84 (0.69) TRPA1AHRGPR84CSNK2A1CYP2A6
SCHEMBL29507011 0.76 GPR84 (0.69) TRPA1AHRGPR84CSNK2A1CYP2A6
SCHEMBL16738736 0.75 EPAS1 (0.49) TRPA1EPAS1HSPB1BRD4
SCHEMBL16738693 0.75 TRPA1 (0.46) TRPA1EPAS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112300154-B Nitrogen-containing heterocyclic compound, preparation method and application thereof 上海弘翊生物科技有限公司 2023-01-24 CN disclosed
CN-112300154-A Nitrogen-containing heterocyclic compound, preparation method and application thereof 上海弘翊生物科技有限公司 2021-02-02 CN disclosed