SCHEMBL28512418

SCHEMBL28512418

O=C(Nc1ccc(F)cc1)C1CCC(n2c(=O)[nH]c3ccccc32)CC1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.58
TSHR P16473 2/20 0.58
PLD2 O14939 4/20 0.55
OPRM1 P35372 3/20 0.54
HTR1A P08908 3/20 0.53
CHRM1 P11229 3/20 0.53
DRD2 P14416 3/20 0.53
HTR2A P28223 3/20 0.53
DRD3 P35462 3/20 0.53
KCNH2 Q12809 3/20 0.53
LMNA P02545 3/20 0.53
MLNR O43193 2/20 0.53
PGR P06401 2/20 0.53
ADRB2 P07550 2/20 0.53
CHRM2 P08172 2/20 0.53
ADRB1 P08588 2/20 0.53
ADRA2A P08913 2/20 0.53
CYP2D6 P10635 2/20 0.53
ADRA2B P18089 2/20 0.53
ADRA2C P18825 2/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22869746 1.00 KMT2A (0.58) KMT2ATSHRPLD2OPRM1HTR1A
SCHEMBL30870137 0.83 KMT2A (0.52) KMT2ATSHRPLD2OPRM1DRD2
SCHEMBL22869512 0.83 KMT2A (0.52) KMT2ATSHRPLD2OPRM1DRD2
SCHEMBL28506714 0.83 KMT2A (0.52) KMT2ATSHRPLD2OPRM1DRD2
SCHEMBL20302481 0.81 ALDH1A1 (0.54) PLD2OPRM1CHRM1LMNACHRM2
SCHEMBL20334166 0.81 ALDH1A1 (0.54) PLD2OPRM1CHRM1LMNACHRM2
SCHEMBL22869573 0.81 HSD11B1 (0.64) PLD2OPRM1LMNAOPRK1PLD1
SCHEMBL22869396 0.81 HTT (0.49) KMT2ATSHRPLD2CHRM1DRD2
SCHEMBL28499858 0.81 HTT (0.49) KMT2ATSHRPLD2CHRM1DRD2
SCHEMBL30870207 0.81 HTT (0.49) KMT2ATSHRPLD2CHRM1DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112074511-A Substituted benzodiazoles and their use in therapy 托马斯·黑勒戴药物研究基金会 2020-12-11 CN claimed
CN-112074511-B Substituted benzodiazoles and their use in therapy 托马斯·黑勒戴药物研究基金会 2024-04-26 CN disclosed