SCHEMBL28514903

SCHEMBL28514903

CN1CCN(c2ccc(-c3cnc4[nH]ccc4n3)cc2C#N)CC1

nearest known ligand 0.51

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 11/20 0.51
DYRK1A Q13627 2/20 0.49
RIPK1 Q13546 1/20 0.46
XDH P47989 1/20 0.45
ROCK2 O75116 2/20 0.45
ROCK1 Q13464 2/20 0.45
CDC42BPB Q9Y5S2 2/20 0.45
TBK1 Q9UHD2 1/20 0.43
JAK2 O60674 2/20 0.42
CDC42BPA Q5VT25 1/20 0.42
CHEK1 O14757 1/20 0.41
JAK3 P52333 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30641871 0.85 MAPK1 (0.54) MAPK1DYRK1ARIPK1JAK2JAK3
SCHEMBL28513749 0.85 MAPK1 (0.54) MAPK1DYRK1ARIPK1JAK2JAK3
SCHEMBL28502428 0.83 RIPK1 (0.54) MAPK1DYRK1ARIPK1XDHROCK2
SCHEMBL28513876 0.83 MAPK1 (0.55) MAPK1DYRK1ARIPK1
SCHEMBL28508679 0.80 MAPK1 (0.59) MAPK1DYRK1ARIPK1CHEK1
SCHEMBL28906226 0.80 ROCK2 (0.47) DYRK1AXDHROCK2ROCK1CDC42BPB
SCHEMBL21590171 0.80 RIPK1 (0.50) MAPK1DYRK1ARIPK1XDHROCK2
SCHEMBL28504401 0.77 MAPK1 (0.55) MAPK1DYRK1ARIPK1JAK2JAK3
SCHEMBL29888818 0.76 MAPK1 (0.56) MAPK1DYRK1ARIPK1
SCHEMBL28769143 0.76 MAPK1 (0.56) MAPK1DYRK1ARIPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112243439-A Pyrrolo [2,3-B ] pyridines or pyrrolo [2,3-B ] pyrazines as HPK1 inhibitors and uses thereof 百济神州有限公司 2021-01-19 CN disclosed