SCHEMBL28513876

SCHEMBL28513876

COc1cc(-c2cnc3[nH]ccc3n2)ccc1N1CCN(C)CC1

nearest known ligand 0.55

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 11/20 0.55
MAP4K1 Q92918 4/20 0.52
DYRK1A Q13627 1/20 0.49
RIPK1 Q13546 1/20 0.46
IL2 P60568 3/20 0.44
MEN1 O00255 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2D6 P10635 1/20 0.43
MAPT P10636 1/20 0.43
KMT2A Q03164 1/20 0.43
TNIK Q9UKE5 2/20 0.42
RPS6KA3 P51812 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28513565 0.88 MAPK1 (0.53) MAPK1MAP4K1DYRK1ARIPK1IL2
SCHEMBL28513749 0.85 MAPK1 (0.54) MAPK1MAP4K1DYRK1ARIPK1
SCHEMBL30641871 0.85 MAPK1 (0.54) MAPK1MAP4K1DYRK1ARIPK1
SCHEMBL28504554 0.83 BRD4 (0.58) MAPK1MAP4K1DYRK1ARIPK1IL2
SCHEMBL28514903 0.83 MAPK1 (0.51) MAPK1DYRK1ARIPK1
SCHEMBL28508679 0.80 MAPK1 (0.59) MAPK1MAP4K1DYRK1ARIPK1MAPT
SCHEMBL28508735 0.80 MAP4K1 (0.61) MAP4K1IL2MEN1CYP1A2CYP2D6
SCHEMBL15542823 0.80 MAPK1 (0.70) MAPK1DYRK1ARIPK1
SCHEMBL29086750 0.78 MAPK1 (0.52) MAPK1MAP4K1DYRK1ARIPK1TNIK
SCHEMBL28504401 0.77 MAPK1 (0.55) MAPK1DYRK1ARIPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112243439-A Pyrrolo [2,3-B ] pyridines or pyrrolo [2,3-B ] pyrazines as HPK1 inhibitors and uses thereof 百济神州有限公司 2021-01-19 CN disclosed