SCHEMBL28516240

SCHEMBL28516240

C=Cc1c(F)cc(B2OC(C)(C)C(C)(C)O2)cc1F.C=Cc1c(F)cc(Br)cc1F

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
LPL P06858 9/20 0.38
LIPG Q9Y5X9 9/20 0.38
ROCK1 Q13464 1/20 0.32
CA1 P00915 3/20 0.31
CA2 P00918 3/20 0.31
CA9 Q16790 3/20 0.31
CA12 O43570 1/20 0.31
CA3 P07451 1/20 0.31
CA4 P22748 1/20 0.31
CA6 P23280 1/20 0.31
CA5A P35218 1/20 0.31
CA7 P43166 1/20 0.31
CA14 Q9ULX7 1/20 0.31
CA5B Q9Y2D0 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21617972 0.92 LPL (0.43) LPLLIPGROCK1CA1CA2
SCHEMBL587344 0.80 LPL (0.39) LPLLIPGROCK1
SCHEMBL23134738 0.79 LPL (0.36) LPLLIPGROCK1CA1CA2
SCHEMBL14488670 0.79 LIPG (0.38) LPLLIPGROCK1CA1CA2
SCHEMBL29016499 0.77 LPL (0.47) LPLLIPGROCK1CA1CA2
SCHEMBL21141913 0.76 ESR1 (0.32)
SCHEMBL4219113 0.76 LPL (0.38) LPLLIPGROCK1
SCHEMBL14488668 0.76 ROCK1 (0.39) LPLLIPGROCK1CA1CA2
SCHEMBL23124209 0.76 LPL (0.43) LPLLIPGROCK1CA1CA2
SCHEMBL21311963 0.74 LPL (0.44) LPLLIPGCA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112334455-B C-mannoside compounds for the treatment of urinary tract infections 葛兰素史密斯克莱知识产权发展有限公司 2022-07-01 CN disclosed
CN-112334455-A C-mannoside compounds for the treatment of urinary tract infections 葛兰素史密斯克莱知识产权发展有限公司 2021-02-05 CN disclosed