SCHEMBL2851771

SCHEMBL2851771

C=C(C(=O)OC)C(O)c1cc(C(=O)O)c(-c2ccccc2)nc1Cl

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 1/20 0.39
ALDH1A1 P00352 1/20 0.37
GABRA1 P14867 1/20 0.35
GABRG2 P18507 1/20 0.35
GABRB3 P28472 1/20 0.35
GABRA5 P31644 1/20 0.35
GABRA3 P34903 1/20 0.35
DHODH Q02127 2/20 0.35
LMNA P02545 1/20 0.35
ATM Q13315 1/20 0.35
KDM4E B2RXH2 3/20 0.35
HPGD P15428 1/20 0.35
HSD17B10 Q99714 1/20 0.35
MAPT P10636 1/20 0.34
KDR P35968 3/20 0.33
PLA2G2A P14555 1/20 0.33
CTSA P10619 2/20 0.33
DGAT1 O75907 1/20 0.33
PPARA Q07869 1/20 0.33
PDE10A Q9Y233 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2849135 0.88 CASP1 (0.56) CASP1ALDH1A1DHODHLMNAATM
SCHEMBL2853119 0.87 CASP1 (0.47) CASP1ALDH1A1DHODHLMNAATM
SCHEMBL2850940 0.87 CASP1 (0.43) CASP1ALDH1A1GABRA1GABRG2GABRB3
SCHEMBL2853071 0.81 CASP1 (0.55) CASP1ALDH1A1LMNAATMKDM4E
SCHEMBL2858064 0.79 CASP1 (0.36) CASP1ALDH1A1DHODHLMNAKDM4E
SCHEMBL2853110 0.78 CASP1 (0.44) CASP1ALDH1A1MAPTCTSADGAT1
SCHEMBL15525179 0.77 EGFR (0.45) CASP1ALDH1A1ATMKDM4EMAPT
SCHEMBL2851268 0.76 CASP1 (0.58) CASP1ALDH1A1DHODHLMNAATM
SCHEMBL13500046 0.75 CASP1 (0.39) CASP1ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL2849381 0.74 CASP1 (0.39) CASP1LMNAKDM4ECTSA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1924558-B1 AN ANTIMALARIAL BAYLIS-HILLMAN ADDUCTS AND A PROCESS FOR THE PREPARATION THEREOF COUNCIL SCIENT IND RES (IN) 2010-01-13 EP claimed