SCHEMBL2858064

SCHEMBL2858064

C=C(C#N)C(O)c1cc(C(=O)O)c(-c2ccccc2)nc1Cl

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 1/20 0.36
KDM4E B2RXH2 5/20 0.35
SMN1; SMN2 Q16637 3/20 0.35
LMNA P02545 3/20 0.35
PDE10A Q9Y233 1/20 0.35
ACMSD Q8TDX5 1/20 0.34
DHODH Q02127 5/20 0.34
ADORA2A P29274 2/20 0.33
ADORA1 P30542 2/20 0.33
ALDH1A1 P00352 5/20 0.33
AKR1C2 P52895 1/20 0.33
AKR1C1 Q04828 1/20 0.33
TDP1 Q9NUW8 3/20 0.32
L3MBTL1 Q9Y468 3/20 0.32
HPGD P15428 2/20 0.32
NPC1 O15118 1/20 0.32
GAA P10253 1/20 0.32
RAB9A P51151 1/20 0.32
EGFR P00533 1/20 0.32
HTT P42858 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2851318 0.85 KDM4E (0.52) CASP1KDM4ESMN1; SMN2LMNADHODH
SCHEMBL2853211 0.83 L3MBTL1 (0.39) KDM4ELMNAPDE10AADORA2AADORA1
SCHEMBL2851771 0.79 CASP1 (0.39) CASP1KDM4ELMNAPDE10ADHODH
SCHEMBL2849135 0.77 CASP1 (0.56) CASP1KDM4ESMN1; SMN2LMNADHODH
SCHEMBL13500074 0.75 SQOR (0.33) KDM4ESMN1; SMN2LMNAPDE10AADORA2A
SCHEMBL2849134 0.74 ALDH1A1 (0.51) KDM4ESMN1; SMN2ALDH1A1TDP1L3MBTL1
SCHEMBL2851215 0.73 KDM4E (0.33) KDM4EACMSDTDP1EGFR
SCHEMBL2853119 0.68 CASP1 (0.47) CASP1KDM4ESMN1; SMN2LMNADHODH
SCHEMBL2850940 0.66 CASP1 (0.43) CASP1LMNAPDE10ADHODHALDH1A1
SCHEMBL2851683 0.66 EGFR (0.30) EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1924558-B1 AN ANTIMALARIAL BAYLIS-HILLMAN ADDUCTS AND A PROCESS FOR THE PREPARATION THEREOF COUNCIL SCIENT IND RES (IN) 2010-01-13 EP claimed