SCHEMBL28517754

SCHEMBL28517754

COC(=O)OCC=Cc1ccc2ccccc2c1

nearest known ligand 0.51

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
APP P05067 1/20 0.51
MAPT P10636 1/20 0.51
HDAC1 Q13547 1/20 0.49
HDAC8 Q9BY41 1/20 0.49
GRIK1 P39086 1/20 0.48
GRIK2 Q13002 1/20 0.48
GRIK3 Q13003 1/20 0.48
NQO2 P16083 2/20 0.48
CNR2 P34972 2/20 0.46
PTGS1 P23219 1/20 0.46
RECQL P46063 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28469494 0.91 PTGS1 (0.51) APPMAPTHDAC1HDAC8GRIK1
SCHEMBL7649080 0.85 PTGS1 (0.49) APPMAPTHDAC1HDAC8GRIK1
SCHEMBL9997162 0.85 PTGS1 (0.49) APPMAPTHDAC1HDAC8GRIK1
SCHEMBL28469496 0.84 RELA (0.51) APPMAPTHDAC1HDAC8GRIK1
SCHEMBL28463082 0.82 CYP3A4 (0.54) MAPTHDAC1HDAC8
SCHEMBL1158016 0.82 MMP1 (0.51)
SCHEMBL1158019 0.82 MMP1 (0.51)
SCHEMBL28706860 0.80 GRIK1 (0.54) MAPTGRIK1GRIK2
SCHEMBL28812360 0.79 TUBB1 (0.44) APPMAPTHDAC1HDAC8PTGS1
SCHEMBL3292230 0.79 GSK3B (0.58) MAPTHDAC1HDAC8GRIK1GRIK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115108938-B Chiral alpha-substituted deuterated amino acid compound and preparation method thereof 武汉大学 2024-04-19 CN disclosed
CN-114736108-B Allyl carbonyl enol compound and synthesis method thereof 同济大学 2023-10-27 CN disclosed
CN-115108938-A Chiral alpha-substituted deuterated amino acid compound and preparation method thereof 武汉大学 2022-09-27 CN disclosed
CN-114736108-A Allyl carbonyl enol compound and synthetic method thereof 同济大学 2022-07-12 CN disclosed
CN-114105822-A Pseudo C2Symmetrical chiral diallyl substituted compound and preparation method and application thereof 武汉大学 2022-03-01 CN disclosed
CN-113861075-A Chiral diallyl substituted compound with three continuous chiral centers and preparation method and application thereof 武汉大学 2021-12-31 CN disclosed
CN-112279770-A Chiral alpha-polysubstituted-alpha-fluorine-containing homoallylamine compound, and preparation method and application thereof 武汉大学 2021-01-29 CN disclosed