SCHEMBL28518544

SCHEMBL28518544

COC(=O)C(C)Cn1cc(Br)cn1

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
OPRK1 P41145 1/20 0.44
HPGD P15428 2/20 0.44
ALDH1A1 P00352 5/20 0.42
LMNA P02545 2/20 0.42
KDM4E B2RXH2 1/20 0.42
ACHE P22303 2/20 0.39
HTT P42858 2/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
KMT2A Q03164 2/20 0.36
MEN1 O00255 1/20 0.36
P2RX3 P56373 1/20 0.36
GAA P10253 2/20 0.36
MGAM O43451 1/20 0.36
SI P14410 1/20 0.36
MGAM2 Q2M2H8 1/20 0.36
MAPT P10636 1/20 0.36
PKM P14618 1/20 0.36
RAB9A P51151 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16029234 0.87 OPRK1 (0.44) OPRK1HPGDALDH1A1LMNAKDM4E
SCHEMBL27696475 0.83 HPGD (0.47) OPRK1HPGDALDH1A1LMNAKDM4E
SCHEMBL18179511 0.82 ACHE (0.42) HPGDALDH1A1LMNAKDM4EACHE
SCHEMBL659599 0.76 HPGD (0.46) OPRK1HPGDALDH1A1LMNAKDM4E
SCHEMBL16912027 0.75 ACHE (0.49) OPRK1HPGDALDH1A1LMNAKDM4E
SCHEMBL1140333 0.74 ALDH1A1 (0.46) HPGDALDH1A1LMNAKDM4EHTT
SCHEMBL18380630 0.74 FFAR1 (0.52) ACHE
SCHEMBL25464716 0.73 OPRK1 (0.43) OPRK1SMN1; SMN2RAB9A
SCHEMBL12993521 0.73 ELANE (0.36) ALDH1A1LMNAKDM4EACHERAB9A
SCHEMBL1581745 0.73 ELANE (0.36) ALDH1A1LMNAKDM4EACHERAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112218857-B P300/CBP HAT inhibitors and methods of use thereof 星座制药公司 2023-11-21 CN disclosed
CN-110678466-B Diazanaphthalenes as HPK1 inhibitors 豪夫迈·罗氏有限公司 2023-01-31 CN disclosed
CN-114450005-A Compounds for the treatment of neurological disorders 星座制药公司 2022-05-06 CN disclosed
CN-112218857-A P300/CBP HAT inhibitors and methods of use thereof 星座制药公司 2021-01-12 CN disclosed