SCHEMBL28518648

SCHEMBL28518648

COc1ccc(Cn2cc3c(n2)CN(C(=O)O)C3)cn1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERCC5 P28715 1/20 0.38
KDR P35968 3/20 0.38
PRMT5 O14744 1/20 0.38
WDR77 Q9BQA1 1/20 0.38
NAMPT P43490 2/20 0.37
MLLT1 Q03111 1/20 0.37
HPGD P15428 1/20 0.37
CYP11B1 P15538 1/20 0.36
TRPV6 Q9H1D0 1/20 0.36
AADAT Q8N5Z0 1/20 0.36
TAS2R14 Q9NYV8 1/20 0.36
PDE1A P54750 1/20 0.36
PDE1B Q01064 1/20 0.36
PDE1C Q14123 1/20 0.36
CACNA1G O43497 1/20 0.36
CACNA1H O95180 1/20 0.36
CACNA1I Q9P0X4 1/20 0.36
TEK Q02763 1/20 0.36
GPR183 P32249 1/20 0.36
ENPP2 Q13822 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22938723 0.86 GPR119 (0.40) KDRAADAT
SCHEMBL28528135 0.84 AADAT (0.51) AADATCACNA1GCACNA1HCACNA1I
SCHEMBL28703394 0.80 SMN1; SMN2 (0.41) AADATCACNA1GCACNA1HCACNA1I
SCHEMBL29774650 0.78 ALDH1A1 (0.43)
SCHEMBL28531542 0.78 ALDH1A1 (0.43)
SCHEMBL28521863 0.78 AADAT (0.54) AADAT
SCHEMBL28507187 0.77 HTT (0.46)
SCHEMBL28527545 0.75 AADAT (0.53) NAMPTAADAT
SCHEMBL28538329 0.75 AADAT (0.38) AADATGPR183
SCHEMBL28525980 0.74 PARP1 (0.39) HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112300167-B Pyrrolopyrazole derivative, preparation method and medical application thereof 上海美迪西生物医药股份有限公司 2022-01-21 CN disclosed
CN-112300167-A Pyrrolopyrazole derivative, preparation method and medical application thereof 上海美迪西生物医药股份有限公司 2021-02-02 CN disclosed