SCHEMBL28518877

SCHEMBL28518877

CN(C)[C@H]1OCCc2ccsc21.O=S(=O)(O)c1ccccc1

nearest known ligand 0.45

Known targets — ChEMBL curated mechanism

BTKCACNA1CCACNA1DCACNA1FCACNA1SCACNA2D1CACNA2D2DRD2GABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQHRH1HTR2AP2RY12

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DRD2 known ✓ P14416 1/20 0.40
HTR2A known ✓ P28223 1/20 0.35
TAAR1 Q96RJ0 9/20 0.45
HTR1A P08908 1/20 0.40
HTR7 P34969 1/20 0.40
TSHR P16473 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
HTR2C P28335 1/20 0.35
KMT2A Q03164 2/20 0.34
NPSR1 Q6W5P4 1/20 0.32
KDM4E B2RXH2 1/20 0.32
MEN1 O00255 1/20 0.32
ALDH1A1 P00352 1/20 0.32
AKR1C3 P42330 2/20 0.32
OPRL1 P41146 1/20 0.32
POLB P06746 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29140412 1.00 TAAR1 (0.45) TAAR1HTR1ADRD2HTR7TSHR
SCHEMBL28517977 0.87 TAAR1 (0.51) TAAR1HTR1ADRD2HTR7
SCHEMBL28511085 0.83 TAAR1 (0.60) TAAR1HTR1ADRD2HTR7
SCHEMBL28511084 0.83 TAAR1 (0.60) TAAR1HTR1ADRD2HTR7
SCHEMBL30733601 0.83 TAAR1 (0.60) TAAR1HTR1ADRD2HTR7
Trifluoromethanesulfonic Acid SCHEMBL28529671 0.83 TAAR1 (0.47) TAAR1HTR1ADRD2HTR7
Hydrochloric Acid SCHEMBL30733605 0.82 TAAR1 (0.59) TAAR1HTR1ADRD2HTR7
Hydrochloric Acid SCHEMBL28522435 0.82 TAAR1 (0.59) TAAR1HTR1ADRD2HTR7
Hydrochloric Acid SCHEMBL29140413 0.82 TAAR1 (0.59) TAAR1HTR1ADRD2HTR7
Hydrochloric Acid SCHEMBL28513760 0.82 TAAR1 (0.59) TAAR1HTR1ADRD2HTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118406063-A Salt, crystal forms and preparation method thereof 赛诺维信制药公司 2024-07-30 CN claimed
CN-118406063-A Salt, crystal forms and preparation method thereof 赛诺维信制药公司 2024-07-30 CN disclosed
CN-112135827-B Salt, crystal forms and preparation method thereof 赛诺维信制药公司 2024-01-12 CN disclosed
CN-112135827-A Salts, crystalline forms and methods for preparing the same 赛诺维信制药公司 2020-12-25 CN disclosed