SCHEMBL28519664

SCHEMBL28519664

Nc1cc(-c2ccccc2)nn1-c1ccc(Br)cc1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 11/20 0.67
RAB9A P51151 10/20 0.67
MEN1 O00255 9/20 0.67
KMT2A Q03164 9/20 0.67
ALDH1A1 P00352 6/20 0.67
TSHR P16473 2/20 0.67
GFER P55789 1/20 0.67
MAPT P10636 10/20 0.63
NPC1 O15118 9/20 0.63
KDM4E B2RXH2 5/20 0.63
STAT1 P42224 1/20 0.63
L3MBTL1 Q9Y468 3/20 0.60
NFKB1 P19838 2/20 0.60
NFKB2 Q00653 2/20 0.60
RELA Q04206 2/20 0.60
CYP1A2 P05177 2/20 0.59
CYP2C19 P33261 2/20 0.59
TP53 P04637 1/20 0.59
CYP3A4 P08684 1/20 0.59
CYP2C9 P11712 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL537890 0.88 RAB9A (0.83) SMN1; SMN2RAB9AMEN1KMT2AALDH1A1
SCHEMBL30229798 0.85 RAB9A (0.84) SMN1; SMN2RAB9AMEN1KMT2AALDH1A1
SCHEMBL28241488 0.84 SMN1; SMN2 (0.74) SMN1; SMN2RAB9AMEN1KMT2AALDH1A1
SCHEMBL28240671 0.84 RAB9A (0.85) SMN1; SMN2RAB9AMEN1KMT2AALDH1A1
SCHEMBL30230060 0.84 SMN1; SMN2 (0.73) SMN1; SMN2RAB9AMEN1KMT2AALDH1A1
SCHEMBL7685096 0.84 USP8 (0.70) SMN1; SMN2RAB9AMEN1KMT2AALDH1A1
SCHEMBL2816383 0.82 USP8 (0.76) RAB9AALDH1A1MAPTNPC1KDM4E
SCHEMBL17619525 0.82 RAB9A (0.69) SMN1; SMN2RAB9AMEN1KMT2AALDH1A1
SCHEMBL30229566 0.80 NPY5R (0.64) SMN1; SMN2RAB9AMEN1KMT2AALDH1A1
SCHEMBL7678240 0.80 NPY5R (0.64) SMN1; SMN2RAB9AMEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114031556-B Synthetic method for preparing 5-amino-N-aryl-3-arylpyrazole compound by green one-pot method 温州大学 2023-03-31 CN disclosed
CN-112300157-B Novel pyrazolopyridine compound with anti-tumor activity and preparation method thereof 烟台大学 2021-08-20 CN disclosed
CN-112300157-A Novel pyrazolopyridine compound with anti-tumor activity and preparation method thereof 烟台大学 2021-02-02 CN disclosed